2.1.1.45 additional information - additional information DHFR inhibition kinetics 742057 2.1.1.45 0.00000006 - D1694 - 485413 2.1.1.45 0.000000095 - methotrexate pH 7.4, 25°C, recombinant enzyme 743569 2.1.1.45 0.000000597 - trimetrexate pH 7.4, 25°C, recombinant enzyme 743569 2.1.1.45 0.000001 - 5-fluoro-2'-deoxyuridylic acid - 485414 2.1.1.45 0.000001 - D1694 pentaglutamate - 485413 2.1.1.45 0.0000015 - D1694 pentaglutamate - 485413 2.1.1.45 0.0000017 - 5-fluoro-2'-deoxyuridylic acid - 485413 2.1.1.45 0.000002 - 5-fluoro-2'-deoxyuridine 5'-monophosphate 22°C 694812 2.1.1.45 0.000002 - 5-fluoro-2'-deoxyuridine 5'-monophosphate inhibited both ThyA and ThyX 694812