5.4.99.5 additional information - oxabicyclic dicarboxylic acid >> 1 mM mutant C88S/R90K 652061 5.4.99.5 0.00032 - (1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid 30°C, pH 7.5, wild-type 651595 5.4.99.5 0.001 - (1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate 30°C, pH 7.5, wild-type 651595 5.4.99.5 0.0023 - (1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate 30°C, pH 7.5, chorismate mutase domain of P-protein 651595 5.4.99.5 0.0028 - chorismate 30°C, pH 7.6, in presence of 0.005 mM tyrosine 651936 5.4.99.5 0.0029 - (1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid 30°C, pH 7.5, mutant DELTA117-127 651595 5.4.99.5 0.003 - oxabicyclic dicarboxylic acid 30°C, pH 7, wild-type 652061 5.4.99.5 0.0037 - 8-hydroxy-2-oxa-bicyclo[3.3.1]non-6-ene-3,5-dicarboxylic acid - 661703 5.4.99.5 0.004 - oxabicyclic dicarboxylic acid 30°C, pH 7, mutant R90G 652061 5.4.99.5 0.0057 - 3-((dihydroxyamino)thio)-4-((3,5-dimethoxyphenethyl)amino)-5-nitrobenzoic acid pH 7.0, 37°C 747259 5.4.99.5 0.0057 - 4-(3,4-dimethoxyphenethylamino)-3-nitro-5-sulfamoylbenzoic acid pH and temperature not specified in the publication 748301 5.4.99.5 0.0057 - 4-[[2-(3,4-dimethoxyphenyl)ethyl]amino]-3-nitro-5-sulfamoylbenzoic acid 4-[[2-(3,4-dimethoxyphenyl)ethyl]amino]-3-nitro-5-sulfamoylbenzoic acid shows the most potent inhibition with Ki value of 0.0057 mM against MtCM 672622 5.4.99.5 0.0076 - (1S,3R,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid 30°C, pH 7.5, chorismate mutase domain of P-protein 651595 5.4.99.5 0.0177 - 2-[2-[3-(tert-butoxycarbonyl)-2-phenyl-1,3-thiazolidin-4-yl]ethyl]-4-methylpentanoic acid pH 7.0, 37°C 747259 5.4.99.5 0.01771 - (2Z)-2-(4-chlorophenyl)-3-(4,5-dimethoxy-2-nitrophenyl)prop-2-enoic acid - 672622 5.4.99.5 0.0211 - (2Z)-2-(4-chlorophenyl)-3-[4-(dimethoxymethyl)-2-nitrophenyl]prop-2-enoic acid pH 7.0, 37°C 747259 5.4.99.5 0.0211 - N-[[3-(tert-butoxycarbonyl)-2-phenyl-1,3-thiazolidin-4-yl]carbonyl]leucine - 672622 5.4.99.5 0.0288 - methyl 4-(methylamino)-3-nitrobenzoate - 672622 5.4.99.5 0.0288 - methyl 4-(methylamino)-3-nitrobenzoate pH 7.0, 37°C 747259 5.4.99.5 0.034 - tyrosine 70°C, pH 7.6 649515 5.4.99.5 0.051 - (1R,3R,5S)-3-carboxy-1-hydroxy-2-oxabicyclo[3.3.1]non-6-ene-5-carboxylate 30°C, pH 7.5, mutant DELTA117-127 651595 5.4.99.5 0.07 - prephenate dimeric chorismate mutase, at 20°C 693664 5.4.99.5 0.17 - prephenate monomeric chorismate mutase, at 20°C 693664 5.4.99.5 0.23 - (1S,3S,5R)-1-hydroxy-5-nitro-2-oxabicyclo[3.3.1]non-6-ene-3-carboxylic acid 30°C, pH 7.5, wild-type 651595 5.4.99.5 1.1 - oxabicyclic dicarboxylic acid 30°C, pH 7, mutant C88K/R90S 652061