3.4.23.47 0.00000016 - TMC-126 - 679179 3.4.23.47 0.00000017 - darunavir - 679179 3.4.23.47 0.00000045 - tipranavir - 679179 3.4.23.47 0.0000006 - saquinavir - 679179 3.4.23.47 0.0000007 - lopinavir - 679179 3.4.23.47 0.0000008 - ritonavir - 679179 3.4.23.47 0.0000012 - (hydroxyethyl)amide isostere - 665102 3.4.23.47 0.0000013 - indinavir - 679179 3.4.23.47 0.0000014 - KNI-764 - 679179 3.4.23.47 0.0000024 - atazanavir - 679179 3.4.23.47 0.0000027 - nelfinavir - 679179 3.4.23.47 0.0000044 - amprenavir - 679179 3.4.23.47 0.000005 - acetyl-pepstatin pH 4.7, competitive versus YVSQNFPIVQNR 665102 3.4.23.47 0.000015 - pepstatin A pH 4.7 665102 3.4.23.47 0.000025 - VSFNF-PSI[CH2-NH]-PQITL pH 5.6, 37°C 644059 3.4.23.47 0.0002 - benzyl (S)-1-((2S,3R)-4-((R)-4-(tert-butylcarbamoyl)thiazolidin-3-yl)-3-hydroxy-1-phenylbutan-2-ylamino)-4-amino-1,4-dioxobutan-2-ylcarbamate pH 4.7, 37°C, synthetic inhibitor 1 644063 3.4.23.47 0.0002 - N-((S)-1-((2S,3R)-4-((3S,4aS,8aS)-3-(tert-butylcarbamoyl)-octahydroisoquinolin-2(1H)-yl)-3-hydroxy-1-phenylbutan-2-ylamino)-4-amino-1,4-dioxobutan-2-yl)quinoline-3-carboxamide pH 4.7, 37°C, synthetic inhibitor 3 644063 3.4.23.47 0.0004 - tert-butyl (2S,3S,5R)-5-(((2S,3R)-3-methyl-1-oxo-1-(phenethylamino)pentan-2-yl)carbamoyl)-1-cyclohexyl-3-hydroxy-6-methylheptan-2-ylcarbamate pH 4.7, 37°C, synthetic inhibitor 5 644063 3.4.23.47 0.0006 - CTLNF-PSI[CH2-NH]-PISP pH 5.6, 37°C 644059 3.4.23.47 0.0007 - (2R,4S,5S)-6-cyclohexyl-5-(3,3-dimethylbutanamido)-4-hydroxy-2-isopropyl-N-((2S,3R)-3-methyl-1-oxo-1-(phenethylamino)pentan-2-yl)hexanamide pH 4.7, 37°C, synthetic inhibitor 4 644063 3.4.23.47 0.04 - darunavir pH 5.6, 37°C 718370 3.4.23.47 0.11 - saquinavir pH 5.6, 37°C 718370 3.4.23.47 0.17 - amprenavir pH 5.6, 37°C 718370