2.7.7.18 additional information - additional information inhibition kinetics, overview 738672 2.7.7.18 0.0079 - K891-0166 pH 7.5, 37°C 727776 2.7.7.18 0.024 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant T12A 738672 2.7.7.18 0.03 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant W117A 738672 2.7.7.18 0.035 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant wild-type enzyme 738672 2.7.7.18 0.037 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant P44A 738672 2.7.7.18 0.056 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant W45A 738672 2.7.7.18 0.094 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant K47A 738672 2.7.7.18 0.114 - 2-(2,4-dimethylphenyl)-N-(4-([(5-methyl-3-isoxazolyl)amino]sulfonyl)phenyl)-4-quinolinecarboxamide pH 7.5, 37°C, recombinant mutant T86A 738672