2.4.2.30 0.001 - suramin 25°C, pH not specified in the publication 722786 2.4.2.30 0.003 - 2-[[3-(dimethylamino)-2-oxopropyl]amino]-5,6-dihydrophenanthridin-6-one wild type enzyme, at pH 7.9 and 22°C 736500 2.4.2.30 0.0041 - N-(acridin-9-yl)-4-nitrobenzamide 25°C, pH not specified in the publication 722786 2.4.2.30 0.0041 - N-[2-oxo-4-(phenylamino)-3,8a-dihydro-2H-chromen-3-yl]acetamide 25°C, pH not specified in the publication 722786 2.4.2.30 0.007 - 8-fluoro-2-[3-(piperidin-1-yl)propanesulfonyl]-1H,2H,3H,4H,5H,6H-benzo[c]1,6-naphthyridin-6-one wild type enzyme, at pH 7.9 and 22°C 736500 2.4.2.30 0.0075 - 2-(4-[4-[(2,4-dimethoxyphenyl)amino]quinazolin-2-yl]piperazin-1-yl)ethanol 25°C, pH not specified in the publication 722786 2.4.2.30 0.00862 - 3-(4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)propanoic acid at pH 7.5 and 22°C 736518 2.4.2.30 0.011 - N-[[1-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]methyl]methanesulfonamide at pH 7.4 and 37°C 736475 2.4.2.30 0.018 - 4-[8-fluoro-6-oxo-1H,2H,3H,4H,5H,6H-benzo[c]1,6-naphthyridin-2-yl]butanoic acid wild type enzyme, at pH 7.9 and 22°C 736500 2.4.2.30 0.019 - 8-fluoro-2-[3-(piperidin-1-yl)propyl]-1H,2H,3H,4H,5H,6H-benzo[c]1,6-naphthyridin-6-one wild type enzyme, at pH 7.9 and 22°C 736500 2.4.2.30 0.024 - 4-[8-fluoro-6-oxo-1H,2H,3H,4H,5H,6H-benzo[c]1,6-naphthyridin-2-yl]butanoic acid wild type enzyme, at pH 7.9 and 22°C 736500 2.4.2.30 0.033 - exosin pH 6.0, 30°C 694800