2.3.1.B41 (4R)-1-[(benzyloxy)carbonyl]-4-hydroxy-L-prolyl-N6-ethanethioyl-N-phenyl-L-lysinamide 0.2 mM, 56% inhibition, substrate: Ac-RYQ(N6-acetyl)K-7-amido-4-methylcoumarin 196340 2.3.1.B41 (9H-fluoren-9-yl)methyl(6-acetamido-1-(dodecylamino)-1-oxohexan-2-yl)carbamate - 245404 2.3.1.B41 (9H-fluoren-9-yl)methyl(6-acetamido-1-(dodecylamino)-1-oxohexanyl) carbamate - 247434 2.3.1.B41 1-(4,5-dihydropyrrolo[1,2-a]quinoxalin-4-yl)naphthalen-2-ol - 245472 2.3.1.B41 1-(tert-butoxycarbonyl)-L-prolyl-N6-ethanethioyl-N-phenyl-L-lysinamide 0.2 mM, 32% inhibition, substrate: Ac-RYQ(N6-acetyl)K-7-amido-4-methylcoumarin 196341 2.3.1.B41 2,4-dioxo-N-(4-(pyridin-3-yloxy)phenyl)-1,2,3,4-tetrahydroquinazoline-6-sulfonamide i.e. compound Q, a SIRT6 inhibitor with quinazolinedione-like structure, which reduces both SIRT6 deacetylase and deacylase activities 247435 2.3.1.B41 2,6-diamino-N-dodecylhexanamide - 245520 2.3.1.B41 2,6-diamino-N-octadecylhexanamide - 245521 2.3.1.B41 2-acetamido-6-amino-N-octadecylhexanamide - 245631 2.3.1.B41 2-acetamido-6-amino-N-tetradecylhexanamide - 247433