4.6.1.12 5-fluorocytidine KD value of 2.02 mM 12387 4.6.1.12 artesunate - 18934 4.6.1.12 Chloroquine - 1439 4.6.1.12 Cidofovir KD value of ca. 40 mM 36543 4.6.1.12 Cytosine arabinoside monophosphate KD value of 18.91 mM 43953 4.6.1.12 EDTA 5 mM. Activity can be restored by the addition of Mg2+ to a concentration of 10 mM 21 4.6.1.12 additional information 5-(1,3-benzodioxol-5-ylamino)-5-oxopentanoic acid, 2-[(2,6-diaminopyrimidin-4-yl)sulfanyl]acetamide and 4-(5-amino-1,3,4-oxadiazol-2-yl)-1,2,5-oxadiazol-3-amine are inactive. Activity with compounds 2-amino-N-hydroxy-acetimidic acid, N-hydroxy-nicotinimidic acid, 5-bromo-thiophene-2-sulfonic acid amide, 4-bromobenzenesulfonamide and 4-(4-dimethylamino-phenylazo)-benzenesulfonamide are not measurable 2 4.6.1.12 N-([4-[(4-amino-2-oxopyrimidin-1(2H)-yl)methyl]-1-naphthyl]methyl)-4-chlorobenzamide 1 mM, 52% inhibition 63523 4.6.1.12 N-([4-[(4-amino-2-oxopyrimidin-1(2H)-yl)methyl]-1-naphthyl]methyl)benzamide 1 mM, 59% inhibition 63522 4.6.1.12 N-[4-[(6-aminopyridin-3-yl)amino]-3-methylbenzyl]-4-(trifluoromethyl)benzamide 1 mM, 60% inhibition 63521