2.6.1.5 2-aminooxyacetate - 172051 2.6.1.5 3,4-dihydroxyphenylalanine - 1782 2.6.1.5 3-(3,4-Dihydroxyphenyl)-2-methylalanine - 29458 2.6.1.5 3-methoxydopamine - 91498 2.6.1.5 3-Methoxytyrosine - 43336 2.6.1.5 Ag2+ - 1041 2.6.1.5 alpha-Methyltyrosine - 43749 2.6.1.5 Ca2+ - 15 2.6.1.5 Canaline - 5532 2.6.1.5 Hg2+ - 33 2.6.1.5 homovanillic acid - 12554 2.6.1.5 L-glutamate - 41 2.6.1.5 Mn2+ - 11 2.6.1.5 normetanephrine - 7260 2.6.1.5 Zn2+ - 14 2.6.1.5 methiozolin 0.5 mM: 91% inhibition of enzyme activity, 0.25 mM: 57% inhibition of enzyme activity 172048 2.6.1.5 cinmethylin 0.5 mM: 96% inhibition of enzyme activity, 0.25 mM: 20% inhibition of enzyme activity 172047 2.6.1.5 EDTA 1 mM, 21% residual activity 21 2.6.1.5 Aminooxyacetate 1 mM, complete inhibition 1374 2.6.1.5 phenylhydrazine 1 mM, complete inhibition 398 2.6.1.5 sodium dodecylsulfate 1 mM, complete inhibition 1066 2.6.1.5 2-chloro-3-(5-{[(2,6-difluorobenzyl)oxy]methyl}-5-methyl-4,5-dihydro-1,2-oxazol-3-yl)-6-(propan-2-yl)pyridine 1 mM: 79% inhibition of enzyme activity, 0.5 mM: 67% inhibition of enzyme activity, 0.25 mM: 44% inhibition of enzyme activity 172050 2.6.1.5 3-(5-{[(2,6-difluorobenzyl)oxy]methyl}-5-methyl-4,5-dihydro-1,2-oxazol-3-yl)pyridine-2-carbonitrile 1 mM: 82% inhibition of enzyme activity, 0.5 mM: 46% inhibition of enzyme activity, 0.25 mM: 8% inhibition of enzyme activity 172049 2.6.1.5 AgNO3 10 mM, complete inhibition 360 2.6.1.5 CuSO4 10 mM, complete inhibition 263 2.6.1.5 kynuric acid 10 mM, complete inhibition 125165 2.6.1.5 SnCl2 10 mM, complete inhibition 3228 2.6.1.5 dopamine 100% inhibition with tyrosine at 3 mM and dopamine at 12 mM 242 2.6.1.5 tyramine 13% inhibition with tyrosine at 3 mM and tyramine at 12 mM 280 2.6.1.5 5-hydroxytryptophan 30% inhibition with tyrosine at 3 mM and 5-hydroxytryptophan at 12 mM 2540 2.6.1.5 phenylacetic acid 30% inhibition with tyrosine at 3 mM and phenylacetic acid at 12 mM 960 2.6.1.5 serotonin 37% inhibition with tyrosine at 3 mM and serotonin at 12 mM 437 2.6.1.5 indole-3-acetic acid 42% inhibition with tyrosine at 3 mM and indole-3-acetic acid at 12 mM 2965 2.6.1.5 Indole-3-propionic acid 48% inhibition with tyrosine at 3 mM and indole-3-propionic acid at 12 mM 6537 2.6.1.5 vanillylmandelic acid 51% inhibition with tyrosine at 3 mM and vanillylmandelic acid at 3 mM 30503 2.6.1.5 5-hydroxyindole acetic acid 55% inhibition with tyrosine at 3 mM and 5-hydroxyindole acetic acid at 12 mM 43544 2.6.1.5 dihydroxymandelic acid 65% inhibition with tyrosine at 3 mM and dihydroxymandelic acid at 3 mM 93201 2.6.1.5 indole-3-butyric acid 71% inhibition with tyrosine at 3 mM and indole-3-butyric acid at 12 mM 12559 2.6.1.5 (4-hydroxyphenyl)acetic acid 74% inhibition with tyrosine at 3 mM and (4-hydroxyphenyl)acetic acid at 12 mM 10446 2.6.1.5 Phenylethylamine 80% inhibition with tyrosine at 3 mM and phenylethylamine at 12 mM 900 2.6.1.5 dihydroxyphenylacetic acid 88% inhibition with tyrosine at 3 mM and dihydroxyphenylacetic acid at 3 mM 29946 2.6.1.5 D-tyrosine 9% inhibition with tyrosine at 3 mM and D-tyrosine at 12 mM 1643 2.6.1.5 L-glutamate competitive inhibition 41 2.6.1.5 norepinephrine competitive inhibition 975 2.6.1.5 Dextran sulfate dextran sulfate inhibits TAT activity but conditioned macrophage medium reliably increases enzyme activity in hepatocytes 2775 2.6.1.5 2-oxoglutarate enzyme shows substrate inhibition 34 2.6.1.5 beta-phenylalanine enzyme shows substrate inhibition 88728 2.6.1.5 homogentisate half-maximal inhibition with 15 micromolar 1826 2.6.1.5 rosmarinic acid isoenzymes TAT-2 and TAT-3 2035 2.6.1.5 Aminooxyacetate probably acts reacting with the cofactor 1374 2.6.1.5 Canaline probably acts reacting with the cofactor 5532 2.6.1.5 4-methylsulfonyl-2,5,6,2',4'-pentachlorobiphenyl significant reduction of dexamethasone-induced activity, 50% inhibition at 0.0007 mM 125166 2.6.1.5 4-methylsulfonyl-2,5,6,2',4',5'-hexachlorobiphenyl significant reduction of dexamethasone-induced activity, 50% inhibition at 0.0008 mM 125167 2.6.1.5 ketoconazole significant reduction of dexamethasone-induced activity, 50% inhibition at 0.0011 mM 483 2.6.1.5 tolylfluanid significant reduction of dexamethasone-induced activity, 50% inhibition at 0.0014 mM 125168 2.6.1.5 3,4-Dihydroxyphenyllactate strong inhibition of all the three TAT isoenzymes 20609 2.6.1.5 2-oxoglutarate substrate inhibition at high concentration 34 2.6.1.5 Urea the enzyme shows a gradual decrease in the activity till 2.5 M urea, after which the complete loss of activity is measured 116 2.6.1.5 D-Aspartate weak inhibition 634 2.6.1.5 alpha-Methyl-L-aspartate with L-tyrosine and 2-oxoglutarate or oxaloacetate as substrates 96130 2.6.1.5 beta-Methyl-L-aspartate with L-tyrosine and 2-oxoglutarate or oxaloacetate as substrates 92777 2.6.1.5 L-aspartate with L-tyrosine and 2-oxoglutarate or oxaloacetate as substrates 97