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Literature summary extracted from

  • Welches, W.R.; Broshihan, K.B.; Ferrario, C.M.
    A comparison of the properties and enzymatic activities of three angiotensin processing enzymes: angiotensin converting enzyme, prolyl endopeptidase and neutral endopeptidase 24.11 (1993), Life Sci., 52, 1461-1480.
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
3.4.24.11
-
Oryctolagus cuniculus

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.24.11 EDTA
-
Bos taurus
3.4.24.11 EDTA
-
Homo sapiens
3.4.24.11 EDTA
-
Mus musculus
3.4.24.11 EDTA
-
Oryctolagus cuniculus
3.4.24.11 EDTA
-
Rattus norvegicus
3.4.24.11 EDTA
-
Sus scrofa
3.4.24.11 NaCl brain enzyme; lung enzyme Mus musculus
3.4.24.11 NaCl no inhibition of the enzyme from brain and kidney Oryctolagus cuniculus
3.4.24.11 NaCl brain enzyme Rattus norvegicus
3.4.24.11 phosphoramidon
-
Homo sapiens
3.4.24.11 phosphoramidon
-
Mus musculus
3.4.24.11 phosphoramidon
-
Rattus norvegicus
3.4.24.11 phosphoramidon
-
Sus scrofa
3.4.24.11 thiol kidney enzyme; lung enzyme Homo sapiens
3.4.24.11 thiol lung enzyme Mus musculus
3.4.24.11 thiol kidney enzyme Oryctolagus cuniculus
3.4.24.11 thiol brain enzyme Rattus norvegicus
3.4.24.11 thiol intestine enzyme; kidney enzyme Sus scrofa
3.4.24.11 thiorphan
-
Homo sapiens
3.4.24.11 thiorphan
-
Mus musculus
3.4.24.11 thiorphan
-
Rattus norvegicus
3.4.24.11 thiorphan
-
Sus scrofa

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.24.11 0.008
-
Tyr-Gly-Gly-Phe-Met
-
Rattus norvegicus
3.4.24.11 0.022
-
Met-enkephalin
-
Homo sapiens
3.4.24.11 0.0319
-
Substance P
-
Sus scrofa
3.4.24.11 0.036
-
angiotensin I
-
Homo sapiens
3.4.24.11 0.039
-
neurotensin
-
Homo sapiens
3.4.24.11 0.04
-
Met-enkephalin
-
Bos taurus
3.4.24.11 0.062
-
Met5-enkephalin
-
Sus scrofa
3.4.24.11 0.074
-
Leu-enkephalin
-
Homo sapiens
3.4.24.11 0.078
-
neurotensin
-
Sus scrofa
3.4.24.11 0.086
-
Leu5-enkephalin
-
Sus scrofa
3.4.24.11 0.092
-
bradykinin
-
Rattus norvegicus
3.4.24.11 0.092
-
bradykinin
-
Sus scrofa
3.4.24.11 0.12
-
bradykinin
-
Oryctolagus cuniculus
3.4.24.11 0.162
-
bradykinin
-
Homo sapiens
3.4.24.11 0.19
-
Substance P
-
Homo sapiens
3.4.24.11 0.755
-
Luteinizing hormone-releasing hormone
-
Rattus norvegicus
3.4.24.11 0.755
-
Luteinizing hormone-releasing hormone
-
Sus scrofa

Organism

EC Number Organism UniProt Comment Textmining
3.4.24.11 Bos taurus
-
-
-
3.4.24.11 Homo sapiens
-
-
-
3.4.24.11 Mus musculus
-
-
-
3.4.24.11 Oryctolagus cuniculus
-
-
-
3.4.24.11 Rattus norvegicus
-
-
-
3.4.24.11 Sus scrofa
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.24.11 kidney
-
Mus musculus
-
3.4.24.11 kidney
-
Homo sapiens
-
3.4.24.11 kidney
-
Rattus norvegicus
-
3.4.24.11 kidney
-
Sus scrofa
-
3.4.24.11 kidney
-
Oryctolagus cuniculus
-
3.4.24.11 lung
-
Rattus norvegicus
-
3.4.24.11 lung
-
Sus scrofa
-
3.4.24.11 testis
-
Rattus norvegicus
-
3.4.24.11 testis
-
Sus scrofa
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.24.11 angiotensin I + H2O
-
Homo sapiens ?
-
?
3.4.24.11 angiotensin I + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 angiotensin I + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O
-
Homo sapiens ?
-
?
3.4.24.11 Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 bradykinin + H2O
-
Homo sapiens ?
-
?
3.4.24.11 bradykinin + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 bradykinin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 bradykinin + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Homo sapiens ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Bos taurus ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 Luteinizing hormone-releasing hormone + H2O
-
Homo sapiens ?
-
?
3.4.24.11 Luteinizing hormone-releasing hormone + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 Luteinizing hormone-releasing hormone + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Luteinizing hormone-releasing hormone + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 neurotensin + H2O
-
Homo sapiens ?
-
?
3.4.24.11 neurotensin + H2O
-
Rattus norvegicus ?
-
?
3.4.24.11 neurotensin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 neurotensin + H2O
-
Oryctolagus cuniculus ?
-
?
3.4.24.11 Substance P + H2O
-
Homo sapiens ?
-
?
3.4.24.11 Substance P + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Homo sapiens Tyr-Gly-Gly + Phe-Met
-
?
3.4.24.11 Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Rattus norvegicus Tyr-Gly-Gly + Phe-Met
-
?
3.4.24.11 Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Sus scrofa Tyr-Gly-Gly + Phe-Met
-
?
3.4.24.11 Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Bos taurus Tyr-Gly-Gly + Phe-Met
-
?

pH Optimum

EC Number pH Optimum Minimum pH Optimum Maximum Comment Organism
3.4.24.11 6
-
kidney enzyme Oryctolagus cuniculus
3.4.24.11 6.5
-
kidney enzyme Homo sapiens
3.4.24.11 6.5 7 brain enzyme Rattus norvegicus
3.4.24.11 7 7.5 kidney enzyme Sus scrofa
3.4.24.11 7
-
-
Mus musculus
3.4.24.11 7
-
-
Rattus norvegicus
3.4.24.11 7
-
intestine Sus scrofa
3.4.24.11 7
-
kidney Homo sapiens
3.4.24.11 8
-
-
Rattus norvegicus