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Literature summary extracted from

  • Landry, C.; Santagata, P.; Bawab, W.; Fournie-Zaluski, M.C.; Roques, B.P.; Vinay, P.; Crine, P.
    Characterization of neutral endopeptidase 24.11 in dog glomeruli (1993), Biochem. J., 291, 773-779.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.24.11 2-[(3-iodohydroxy)phenylmethyl]-4-N-[3-hydroxyamino-3-oxo-1-phenylmethylpropyl]-amino-4-oxobutanoic acid i.e. RB104, highly selective and potent inhibitor Canis lupus familiaris
3.4.24.11 phosphoramidon
-
Canis lupus familiaris
3.4.24.11 thiorphan
-
Canis lupus familiaris

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.24.11 0.07
-
D-Ala2-Leu5-enkephalin enzyme from tubules Canis lupus familiaris
3.4.24.11 0.076
-
D-Ala2-Leu5-enkephalin enzyme from glomeruli Canis lupus familiaris

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.4.24.11 membrane glomerular enzyme is membrane-bound Canis lupus familiaris 16020
-

Molecular Weight [Da]

EC Number Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
3.4.24.11 94000
-
x * 94000, enzyme from tubules, SDS-PAGE Canis lupus familiaris
3.4.24.11 104000
-
x * 104000, enzyme from glomeruli, SDS-PAGE Canis lupus familiaris

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.4.24.11 additional information Canis lupus familiaris the enzyme may play an important role as regulator of plasma-derived peptides in the nephron ?
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.4.24.11 Canis lupus familiaris
-
-
-

Posttranslational Modification

EC Number Posttranslational Modification Comment Organism
3.4.24.11 side-chain modification glycoprotein Canis lupus familiaris

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.24.11 kidney glomeruli, tubules Canis lupus familiaris
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.24.11 D-Ala2-Leu5-enkephalin + H2O i.e. Tyr-D-Ala-Gly-Phe-Leu Canis lupus familiaris Tyr-D-Ala-Gly + Phe-Leu
-
?
3.4.24.11 additional information the enzyme may play an important role as regulator of plasma-derived peptides in the nephron Canis lupus familiaris ?
-
?

Subunits

EC Number Subunits Comment Organism
3.4.24.11 ? x * 94000, enzyme from tubules, SDS-PAGE Canis lupus familiaris
3.4.24.11 ? x * 104000, enzyme from glomeruli, SDS-PAGE Canis lupus familiaris

Turnover Number [1/s]

EC Number Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
3.4.24.11 19
-
D-Ala2-Leu5-enkephalin enzyme from tubules Canis lupus familiaris
3.4.24.11 20.7
-
D-Ala2-Leu5-enkephalin enzyme from glomeruli Canis lupus familiaris