EC Number | Cloned (Comment) | Organism |
---|---|---|
3.4.24.11 | cloned into the pQE expression vector, resulting in the fusion of a hexahistidine at the N-terminus, expression in Escherichia coli | Lactococcus lactis |
EC Number | Protein Variants | Comment | Organism |
---|---|---|---|
3.4.24.11 | E535Q | inactive enzyme | Lactococcus lactis |
3.4.24.11 | H587Q | inactive enzyme | Lactococcus lactis |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.11 | diethyl dicarbonate | - |
Lactococcus lactis | |
3.4.24.11 | phosphoramidon | - |
Lactococcus lactis | |
3.4.24.11 | thiorphan | weak | Lactococcus lactis |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.11 | 0.0004 | - |
angiotensin I | - |
Lactococcus lactis | |
3.4.24.11 | 0.0018 | - |
Vasoactive intestinal peptide | - |
Lactococcus lactis | |
3.4.24.11 | 0.0028 | - |
adrenocorticotropic hormone | - |
Lactococcus lactis | |
3.4.24.11 | 0.005 | - |
bradykinin | - |
Lactococcus lactis | |
3.4.24.11 | 0.00654 | - |
beta-endorphin | - |
Lactococcus lactis | |
3.4.24.11 | 0.0082 | - |
dynorphin A-17 | - |
Lactococcus lactis | |
3.4.24.11 | 0.01 | - |
Substance P | - |
Lactococcus lactis | |
3.4.24.11 | 0.01 | - |
dynorphin A-13 | - |
Lactococcus lactis | |
3.4.24.11 | 0.025 | - |
dynorphin A-6 | - |
Lactococcus lactis | |
3.4.24.11 | 0.035 | - |
dynorphin A-10 | - |
Lactococcus lactis | |
3.4.24.11 | 0.04 | - |
dynorphin A-9 | - |
Lactococcus lactis | |
3.4.24.11 | 0.1 | - |
Met-enkephalin | - |
Lactococcus lactis | |
3.4.24.11 | 0.135 | - |
alpha-neoendorphin | - |
Lactococcus lactis | |
3.4.24.11 | 0.2 | - |
Leu-enkephalin | - |
Lactococcus lactis | |
3.4.24.11 | 0.298 | - |
dynorphin A-8 | - |
Lactococcus lactis | |
3.4.24.11 | 0.41 | - |
Met-enkephalin amide | - |
Lactococcus lactis | |
3.4.24.11 | 0.612 | - |
Leu-enkephalinamide | - |
Lactococcus lactis |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.24.11 | Lactococcus lactis | - |
- |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
3.4.24.11 | - |
Lactococcus lactis |
EC Number | Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|---|
3.4.24.11 | 0.203 | - |
cleavage of succinyl-Arg-Pro-Phe-His-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide | Lactococcus lactis |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.24.11 | adrenocorticotropic hormone + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | alpha-neoendorphin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | angiotensin I + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | beta-endorphin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | beta-neoendorphin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | bradykinin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin + H2O | dynorphin A-6, A-8, A-9, A-10, A-13 and A-17 | Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-10 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-13 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-17 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-6 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-8 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | dynorphin A-9 + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | enkephalin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Leu-enkephalin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Leu5-enkephalinamide + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Met-enkephalin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Met-enkephalin amide + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Substance P + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | succinyl-Arg-Pro-Phe-His-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin + H2O | - |
Lactococcus lactis | ? | - |
? | |
3.4.24.11 | Vasoactive intestinal peptide + H2O | - |
Lactococcus lactis | ? | - |
? |
EC Number | Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.11 | 0.5 | - |
Met-enkephalin amide | - |
Lactococcus lactis | |
3.4.24.11 | 1.7 | - |
adrenocorticotropic hormone | - |
Lactococcus lactis | |
3.4.24.11 | 1.8 | - |
Vasoactive intestinal peptide | - |
Lactococcus lactis | |
3.4.24.11 | 4.3 | - |
bradykinin | - |
Lactococcus lactis | |
3.4.24.11 | 7.8 | - |
Met-enkephalin | - |
Lactococcus lactis | |
3.4.24.11 | 8.2 | - |
Leu-enkephalinamide | - |
Lactococcus lactis | |
3.4.24.11 | 14 | - |
dynorphin A-6 | - |
Lactococcus lactis | |
3.4.24.11 | 15 | - |
Leu-enkephalin | - |
Lactococcus lactis | |
3.4.24.11 | 18.6 | - |
dynorphin A-13 | - |
Lactococcus lactis | |
3.4.24.11 | 19.6 | - |
dynorphin A-8 | - |
Lactococcus lactis | |
3.4.24.11 | 23.8 | - |
dynorphin A-10 | - |
Lactococcus lactis | |
3.4.24.11 | 25.4 | - |
dynorphin A-17 | - |
Lactococcus lactis | |
3.4.24.11 | 26 | - |
beta-endorphin | - |
Lactococcus lactis | |
3.4.24.11 | 28 | - |
Substance P | - |
Lactococcus lactis | |
3.4.24.11 | 32.2 | - |
dynorphin A-9 | - |
Lactococcus lactis | |
3.4.24.11 | 44.6 | - |
alpha-neoendorphin | - |
Lactococcus lactis |