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Literature summary extracted from

  • Kenny, A.J.; Bowes, M.A.; Gee, N.S.; Matsas, R.
    Endopeptidase-24.11: a cell-surface enzyme for metabolizing regulatory peptides (1985), Biochem. Soc. Trans., 13, 293-295.
    View publication on PubMed

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.24.11 0.032
-
Substance P
-
Sus scrofa
3.4.24.11 0.039
-
Met5-enkephalin-Arg6
-
Sus scrofa
3.4.24.11 0.05
-
Met5-enkephalin-Arg6Phe7
-
Sus scrofa
3.4.24.11 0.062
-
Met5-enkephalin
-
Sus scrofa
3.4.24.11 0.086
-
Leu5-enkephalin
-
Sus scrofa
3.4.24.11 0.088
-
D-Ala2-Leu5-enkephalin
-
Sus scrofa
3.4.24.11 0.092
-
bradykinin
-
Sus scrofa
3.4.24.11 0.106
-
Physalaemin
-
Sus scrofa
3.4.24.11 0.111
-
Leu5-enkephalin-Arg6
-
Sus scrofa
3.4.24.11 0.119
-
dynorphin(1-9)
-
Sus scrofa
3.4.24.11 0.296
-
cholecystokinin-8
-
Sus scrofa
3.4.24.11 0.432
-
D-Ala2-Met5-enkephalinamide
-
Sus scrofa
3.4.24.11 0.68
-
Leu5-enkephalinamide
-
Sus scrofa
3.4.24.11 0.773
-
D-Ala2-Leu5-enkephalinamide
-
Sus scrofa

Organism

EC Number Organism UniProt Comment Textmining
3.4.24.11 Sus scrofa
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.24.11 central nervous system
-
Sus scrofa
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.24.11 Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O
-
Sus scrofa ?
-
?
3.4.24.11 bradykinin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 cholecystokinin-8 + H2O
-
Sus scrofa ?
-
?
3.4.24.11 D-Ala2-Leu5-enkephalin + H2O i.e. Tyr-D-Ala-Gly-Phe-Leu Sus scrofa Tyr-D-Ala-Gly + Phe-Leu
-
?
3.4.24.11 D-Ala2-Leu5-enkephalinamide + H2O
-
Sus scrofa ?
-
?
3.4.24.11 dynorphin(1-9) + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Leu5-enkephalin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Leu5-enkephalin-Arg6 + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Leu5-enkephalinamide + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Met5-enkephalin-Arg6-Phe7 + H2O
-
Sus scrofa ?
-
?
3.4.24.11 physalaemin + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Substance P + H2O
-
Sus scrofa ?
-
?
3.4.24.11 Tyr-D-Ala-Gly-Phe-Met + H2O
-
Sus scrofa Tyr-D-Ala-Gly + Phe-Met
-
?
3.4.24.11 Tyr-D-Ala-Gly-Phe-Met-NH2 + H2O
-
Sus scrofa Tyr-D-Ala-Gly + Phe-Met-NH2
-
?
3.4.24.11 Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Sus scrofa Tyr-Gly-Gly + Phe-Met
-
?