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Literature summary extracted from

  • Araujo, N.A.; Rincon, M.; Vonasek, E.; Calabokis, M.; Bubis, J.
    Biochemical characterization of the cAMP-dependent protein kinase regulatory subunit-like protein from Trypanosoma equiperdum, detection of its inhibitory activity, and identification of potential interacting proteins (2020), Biochimie, 168, 110-123 .
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.11.11 Trypanosoma equiperdum PKA regulatory subunit-like protein uncompetitive or anticompetitive inhibitor Sus scrofa

Organism

EC Number Organism UniProt Comment Textmining
2.7.11.11 Sus scrofa
-
-
-
2.7.11.11 Trypanosoma equiperdum A0A068EPY7 protein kinase A regulatory subunit
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
2.7.11.11 heart
-
Sus scrofa
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2.7.11.11 ATP + Kemptide
-
Sus scrofa ADP + phosphorylated Kemptide
-
?

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
2.7.11.11 0.00117
-
Trypanosoma equiperdum PKA regulatory subunit-like protein pH and temperature not specified in the publication Sus scrofa