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Literature summary extracted from

  • Teraoka, Y.; Kume, S.; Lin, Y.; Atsuji, S.; Inui, T.
    Comprehensive evaluation of the binding of lipocalin-type prostaglandin D synthase to poorly water-soluble drugs (2017), Mol. Pharm., 14, 3558-3567 .
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
5.3.99.2 expressed in Escherichia coli BL21(DE3) cells Homo sapiens

Protein Variants

EC Number Protein Variants Comment Organism
5.3.99.2 C65A/C167A inactive Homo sapiens

Inhibitors

EC Number Inhibitors Comment Organism Structure
5.3.99.2 atovaquone
-
Homo sapiens
5.3.99.2 imatinib
-
Homo sapiens
5.3.99.2 lapatinib
-
Homo sapiens
5.3.99.2 nilotinib
-
Homo sapiens
5.3.99.2 telmisartan
-
Homo sapiens

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
5.3.99.2 Prostaglandin H2 Homo sapiens
-
Prostaglandin D2
-
?

Organism

EC Number Organism UniProt Comment Textmining
5.3.99.2 Homo sapiens P41222
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
5.3.99.2 glutathione Sepharose column chromatography and Superdex 75 gel filtration Homo sapiens

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
5.3.99.2 Prostaglandin H2
-
Homo sapiens Prostaglandin D2
-
?

Synonyms

EC Number Synonyms Comment Organism
5.3.99.2 L-PGDS
-
Homo sapiens
5.3.99.2 lipocalin-type prostaglandin d synthase
-
Homo sapiens