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Literature summary extracted from

  • Fallatah, O.; Georges, E.
    Apigenin-induced ABCC1-mediated efflux of glutathione from mature erythrocytes inhibits the proliferation of Plasmodium falciparum (2017), Int. J. Antimicrob. Agents, 50, 673-677 .
    View publication on PubMed

Activating Compound

EC Number Activating Compound Comment Organism Structure
7.6.2.3 apigenin
-
Homo sapiens

Inhibitors

EC Number Inhibitors Comment Organism Structure
7.6.2.3 MK571
-
Homo sapiens

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
7.6.2.3 ATP + H2O + S-(calcein-AM)glutathione[side 1] Homo sapiens
-
ADP + phosphate + S-(calcein-AM)glutathione[side 2]
-
?

Organism

EC Number Organism UniProt Comment Textmining
7.6.2.3 Homo sapiens P08183
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
7.6.2.3 erythrocyte
-
Homo sapiens
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
7.6.2.3 ATP + H2O + S-(calcein-AM)glutathione[side 1]
-
Homo sapiens ADP + phosphate + S-(calcein-AM)glutathione[side 2]
-
?

Subunits

EC Number Subunits Comment Organism
7.6.2.3 ? x * 200000, SDS-PAGE Homo sapiens

Synonyms

EC Number Synonyms Comment Organism
7.6.2.3 ABCC1
-
Homo sapiens
7.6.2.3 MRP1
-
Homo sapiens
7.6.2.3 multidrug resistance-associated protein
-
Homo sapiens

General Information

EC Number General Information Comment Organism
7.6.2.3 physiological function enzyme-mediated efflux of glutathione from mature erythrocytes inhibits the proliferation of Plasmodium falciparum Homo sapiens