EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
7.6.2.2 | amlodipine | - |
Homo sapiens | |
7.6.2.2 | atorvastatin | - |
Homo sapiens | |
7.6.2.2 | azithromycin | - |
Homo sapiens | |
7.6.2.2 | cyclosporin A | - |
Homo sapiens | |
7.6.2.2 | dexniguldipine | - |
Homo sapiens | |
7.6.2.2 | dipyridamole | - |
Homo sapiens | |
7.6.2.2 | Disulfiram | - |
Homo sapiens | |
7.6.2.2 | elacridar | - |
Homo sapiens | |
7.6.2.2 | fumitremorgin C | - |
Homo sapiens | |
7.6.2.2 | Furosemide | - |
Homo sapiens | |
7.6.2.2 | GF120918 | - |
Homo sapiens | |
7.6.2.2 | glibenclamide | - |
Homo sapiens | |
7.6.2.2 | LY335979 | - |
Homo sapiens | |
7.6.2.2 | LY475776 | - |
Homo sapiens | |
7.6.2.2 | MK-571 | - |
Homo sapiens | |
7.6.2.2 | MS-209 | - |
Homo sapiens | |
7.6.2.2 | nifedipine | - |
Homo sapiens | |
7.6.2.2 | novobiocin | - |
Homo sapiens | |
7.6.2.2 | OC144-093 | - |
Homo sapiens | |
7.6.2.2 | ortataxel | - |
Homo sapiens | |
7.6.2.2 | pluronic L61 | - |
Homo sapiens | |
7.6.2.2 | probenecid | - |
Homo sapiens | |
7.6.2.2 | PSC-833 | - |
Homo sapiens | |
7.6.2.2 | quinidine | - |
Homo sapiens | |
7.6.2.2 | R101933 | - |
Homo sapiens | |
7.6.2.2 | reserpine | - |
Homo sapiens | |
7.6.2.2 | ritonavir | - |
Homo sapiens | |
7.6.2.2 | S9788 | - |
Homo sapiens | |
7.6.2.2 | tariquidar | - |
Homo sapiens | |
7.6.2.2 | V-104 | - |
Homo sapiens | |
7.6.2.2 | verapamil | - |
Homo sapiens | |
7.6.2.2 | VX-710 | - |
Homo sapiens | |
7.6.2.2 | XR-9576 | - |
Homo sapiens |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
7.6.2.2 | plasma membrane | - |
Homo sapiens | 5886 | - |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
7.6.2.2 | ATP + H2O + xenobiotic[side 1] | Homo sapiens | - |
ADP + phosphate + xenobiotic[side 2] | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
7.6.2.2 | Homo sapiens | - |
- |
- |
7.6.2.2 | Homo sapiens | P08183 | - |
- |
7.6.2.2 | Homo sapiens | Q2M3G0 | - |
- |
7.6.2.2 | Homo sapiens | Q92887 | - |
- |
7.6.2.2 | Homo sapiens | Q9UNQ0 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
7.6.2.2 | brain | - |
Homo sapiens | - |
7.6.2.2 | brain capillary endothelial cell line | - |
Homo sapiens | - |
7.6.2.2 | culture condition:CD4+ cell | - |
Homo sapiens | - |
7.6.2.2 | enterocyte | - |
Homo sapiens | - |
7.6.2.2 | gall bladder | - |
Homo sapiens | - |
7.6.2.2 | hepatocyte | - |
Homo sapiens | - |
7.6.2.2 | intestinal mucosa | - |
Homo sapiens | - |
7.6.2.2 | intestine | - |
Homo sapiens | - |
7.6.2.2 | kidney | - |
Homo sapiens | - |
7.6.2.2 | liver | - |
Homo sapiens | - |
7.6.2.2 | lymphocyte | - |
Homo sapiens | - |
7.6.2.2 | placenta | - |
Homo sapiens | - |
7.6.2.2 | renal proximal tubule epithelial cell | - |
Homo sapiens | - |
7.6.2.2 | small intestine | - |
Homo sapiens | - |
7.6.2.2 | trophoblast | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
7.6.2.2 | ATP + H2O + 4-aminohippurate[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + 4-aminohippurate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + 5-fluorouracil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + 5-fluorouracil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + actinomycin D[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + actinomycin D[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + adevovir[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + adevovir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + amiodarone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + amiodarone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ampicillin[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + ampicillin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + amprenavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + amprenavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + asimadoline[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + asimadoline[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + azidopine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + azidopine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + azidothymidine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + azidothymidine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + azithromycin[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + azithromycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + BCECF-acetoxymethylester[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + BCECF-acetoxymethylester[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + bepridil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + bepridil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + bisantrene[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + bisantrene[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + calcein acetoxymethylester[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + calcein acetoxymethylester[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + calcein-acetoxymethylester[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + calcein-acetoxymethylester[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cefodizime[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + cefodizime[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cefoperazone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + cefoperazone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ceftriaxone[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + ceftriaxone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ceftriaxone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + ceftriaxone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cerivastatin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + cerivastatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + chlorambucil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + chlorambucil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + chlorpromazine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + chlorpromazine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + chrysin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + chrysin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cidofovir[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + cidofovir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cimetidine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + cimetidine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ciprofloxacin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + ciprofloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cisplatin[side 1] | substrate for P-glycoprotein and MPR2 | Homo sapiens | ADP + phosphate + cisplatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + clarithromycin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + clarithromycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + colchicine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + colchicine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cyclosporin A[side 1] | substrate for P-glycoprotein and BCRP | Homo sapiens | ADP + phosphate + cyclosporin A[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cyclosporin H[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + cyclosporin H[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cytarabine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + cytarabine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + daunorubicin[side 1] | substrate for P-glycoprotein and BCRP | Homo sapiens | ADP + phosphate + daunorubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + delavirdine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + delavirdine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + digoxin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + digoxin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + diltiazem[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + diltiazem[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + docetaxel[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + docetaxel[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + doxorubicin[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + doxorubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + doxycycline[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + doxycycline[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + endosulfan[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + endosulfan[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + epirubicin[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + epirubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + erythromycin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + erythromycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ethinylestradiol-3-O-glucuronide[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + ethinylestradiol-3-O-glucuronide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + etoposide[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + etoposide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + felodipine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + felodipine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + fentanyl[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + fentanyl[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + fexofenadine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + fexofenadine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + FK506[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + FK506[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + gefitinib[side 1] | substrate for P-glycoprotein and BCRP | Homo sapiens | ADP + phosphate + gefitinib[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + genistein-7-glucoside[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + genistein-7-glucoside[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + gramicidin A[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + gramicidin A[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + gramicidin D[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + gramicidin D[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + grepafloxacine[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + grepafloxacine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + grepafloxacin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + grepafloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + Hoechst 33342[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + Hoechst 33342[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + hydroxyurea[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + hydroxyurea[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + imatinib[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + imatinib[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + indinavir[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + indinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + indinavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + indinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + irinotecan[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + irinotecan[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + itraconazole[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + itraconazole[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ketoconazole[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + ketoconazole[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + lamivudine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + lamivudine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + leupeptin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + leupeptin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + levofloxacin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + levofloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + lidocaine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + lidocaine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + lopinavir[side 1] | substrate for MPR2 and BCRP | Homo sapiens | ADP + phosphate + lopinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + lopinavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + lopinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + lovastatin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + lovastatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + methotrexate[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + methotrexate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + methyl parathion[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + methyl parathion[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + mitomycin C[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + mitomycin C[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + mitoxantrone[side 1] | substrate for P-glycoprotein, BCRP, and MPR2 | Homo sapiens | ADP + phosphate + mitoxantrone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + morphine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + morphine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nelfinavir[side 1] | substrate for MPR2 and BCRP | Homo sapiens | ADP + phosphate + nelfinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nelfinavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + nelfinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nicardipine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + nicardipine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nifedipine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + nifedipine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nisoldipine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + nisoldipine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + nitrendipine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + nitrendipine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + norfloxacin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + norfloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ofloxacin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + ofloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + olmesartan[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + olmesartan[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ortataxel[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + ortataxel[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + paraquat[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + paraquat[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + pentazocine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + pentazocine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + pepstatin A[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + pepstatin A[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + phenothiazine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + phenothiazine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + phloridzin[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + phloridzin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + pravastatin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + pravastatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + propafenone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + propafenone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + quercetin 4'-beta-glucoside[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + quercetin 4'-beta-glucoside[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + quercetin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + quercetin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + quinidine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + quinidine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ranitidine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + ranitidine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + reserpine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + reserpine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + rhodamine 123[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + rhodamine 123[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + rifampicin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + rifampicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ritonavir[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + ritonavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ritonavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + ritonavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + rosuvastatin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + rosuvastatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + saquinavir[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + saquinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + saquinavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + saquinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + simvastatin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + simvastatin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + sirolimus[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + sirolimus[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + SN-38[side 1] | substrate for MPR2 and BCRP | Homo sapiens | ADP + phosphate + SN-38[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + sparfloxacin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + sparfloxacin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + tacrolimus[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + tacrolimus[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + tamoxifen[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + tamoxifen[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + temocaprilate[side 1] | substrate for MPR2 | Homo sapiens | ADP + phosphate + temocaprilate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + teniposide[side 1] | substrate for P-glycoprotein and BCRP | Homo sapiens | ADP + phosphate + teniposide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + terfenadine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + terfenadine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + tetracycline[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + tetracycline[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + tiapamil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + tiapamil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + topotecan[side 1] | substrate for P-glycoprotein and BCRP | Homo sapiens | ADP + phosphate + topotecan[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + trans-flupentixol[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + trans-flupentixol[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + trifluoperazine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + trifluoperazine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + valinomycin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + valinomycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + valspodar[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + valspodar[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + verapamil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + verapamil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + vinblastine[side 1] | substrate for P-glycoprotein and MPR2 | Homo sapiens | ADP + phosphate + vinblastine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + vincristine[side 1] | substrate for P-glycoprotein and MPR2 | Homo sapiens | ADP + phosphate + vincristine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + xenobiotic[side 1] | - |
Homo sapiens | ADP + phosphate + xenobiotic[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + zidovudine[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + zidovudine[side 2] | - |
? |
EC Number | Subunits | Comment | Organism |
---|---|---|---|
7.6.2.2 | ? | x * 170000, P-glycoprotein , SDS-PAGE | Homo sapiens |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
7.6.2.2 | ABCB1 | - |
Homo sapiens |
7.6.2.2 | ABCC2 | - |
Homo sapiens |
7.6.2.2 | ABCG2 | - |
Homo sapiens |
7.6.2.2 | BCRP | - |
Homo sapiens |
7.6.2.2 | breast cancer resistance protein | - |
Homo sapiens |
7.6.2.2 | canalicular multispecific organic anion transporter | - |
Homo sapiens |
7.6.2.2 | MDR-ABC transporter | - |
Homo sapiens |
7.6.2.2 | MOAT | - |
Homo sapiens |
7.6.2.2 | MRP2 | - |
Homo sapiens |
7.6.2.2 | multidrug resistance-associated protein 2 | - |
Homo sapiens |
7.6.2.2 | P-glycoprotein | - |
Homo sapiens |
7.6.2.2 | P-gp | - |
Homo sapiens |