Literature summary extracted from

Park, C.H.; Lee, J.H.; Lee, M.Y.; Lee, J.H.; Lee, B.H.; Oh, K.S.
A novel role of G protein-coupled receptor kinase 5 in urotensin II-stimulated cellular hypertrophy in H9c2UT cells (2016), Mol. Cell. Biochem., 422, 151-160.

Inhibitors

EC Number	Inhibitors	Comment	Organism	Structure
2.7.11.16	amlexanox	selective inhibitor	Rattus norvegicus

Organism

EC Number	Organism	UniProt	Comment	Textmining
2.7.11.16	Rattus norvegicus	Q62833	-	-

Source Tissue

EC Number	Source Tissue	Comment	Organism	Textmining
2.7.11.16	cardiomyocyte	-	Rattus norvegicus	-
2.7.11.16	H9c2 cell	-	Rattus norvegicus	-

Synonyms

EC Number	Synonyms	Comment	Organism
2.7.11.16	G protein-coupled receptor kinase 5	-	Rattus norvegicus
2.7.11.16	GRK5	-	Rattus norvegicus

General Information

EC Number	General Information	Comment	Organism
2.7.11.16	physiological function	the enzyme plays a role in urotensin II-mediated cellular hypertrophy via activation of nuclear factor-kappaB and histone deacetylase 5	Rattus norvegicus

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Release 2023.1 (January 2023)