Data extracted from this reference:
Cloned(Commentary)
2.4.2.12
expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL
Mus musculus
Inhibitors
2.4.2.12
(4',5,7-trihydroxyflavone)-(3'->8)-(4',5,7-trihydroxyflavone)
Mus musculus
2.4.2.12
(4',7-dimethoxy-5-hydroxyflavone)-(3'->8)-(4',7-dimethoxy-5-hydroxyflavone)
Mus musculus
2.4.2.12
FK-866
i.e. (2E)-N-[4-(1-benzoylpiperidin-4-yl)butyl]-3-phenylprop-2-enamide
Mus musculus
2.4.2.12
gallotanine
i.e. (2R,3S,5R,6S)-tetrahydro-2H-pyran-2,3,4,5,6-pentaylpentakis(oxycarbonyl-5,6-dihydroxybenzene-3,1-diyl) pentakis(3,4,5-trihydroxybenzoate)
Mus musculus
Organism
Purification (Commentary)
2.4.2.12
immobilized metal ion affinity chromatography
Mus musculus
Substrates and Products (Substrate)
2.4.2.12
nicotinamide + 5-phosphoribosyl 1-diphosphate
721273
Mus musculus
nicotinamide mononucleotide + diphosphate
?
Synonyms
2.4.2.12
nicotinamide phosphoribosyltransferase
Mus musculus
2.4.2.12
PBEF
Mus musculus
2.4.2.12
Visfatin
Mus musculus
IC50 Value
2.4.2.12
0.0000009
i.e. (2E)-N-[4-(1-benzoylpiperidin-4-yl)butyl]-3-phenylprop-2-enamide, pH 7.5, 37°C
Mus musculus
FK-866
2.4.2.12
0.0013
i.e. (2R,3S,5R,6S)-tetrahydro-2H-pyran-2,3,4,5,6-pentaylpentakis(oxycarbonyl-5,6-dihydroxybenzene-3,1-diyl) pentakis(3,4,5-trihydroxybenzoate), pH 7.5, 37°C
Mus musculus
gallotanine
2.4.2.12
0.0066
pH 7.5, 37°C
Mus musculus
(4',5,7-trihydroxyflavone)-(3'->8)-(4',5,7-trihydroxyflavone)
2.4.2.12
0.0175
pH 7.5, 37°C
Mus musculus
(4',7-dimethoxy-5-hydroxyflavone)-(3'->8)-(4',7-dimethoxy-5-hydroxyflavone)
Cloned(Commentary) (protein specific)
2.4.2.12
expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL
Mus musculus
IC50 Value (protein specific)
2.4.2.12
0.0000009
i.e. (2E)-N-[4-(1-benzoylpiperidin-4-yl)butyl]-3-phenylprop-2-enamide, pH 7.5, 37°C
Mus musculus
FK-866
2.4.2.12
0.0013
i.e. (2R,3S,5R,6S)-tetrahydro-2H-pyran-2,3,4,5,6-pentaylpentakis(oxycarbonyl-5,6-dihydroxybenzene-3,1-diyl) pentakis(3,4,5-trihydroxybenzoate), pH 7.5, 37°C
Mus musculus
gallotanine
2.4.2.12
0.0066
pH 7.5, 37°C
Mus musculus
(4',5,7-trihydroxyflavone)-(3'->8)-(4',5,7-trihydroxyflavone)
2.4.2.12
0.0175
pH 7.5, 37°C
Mus musculus
(4',7-dimethoxy-5-hydroxyflavone)-(3'->8)-(4',7-dimethoxy-5-hydroxyflavone)
Inhibitors (protein specific)
2.4.2.12
(4',5,7-trihydroxyflavone)-(3'->8)-(4',5,7-trihydroxyflavone)
Mus musculus
2.4.2.12
(4',7-dimethoxy-5-hydroxyflavone)-(3'->8)-(4',7-dimethoxy-5-hydroxyflavone)
Mus musculus
2.4.2.12
FK-866
i.e. (2E)-N-[4-(1-benzoylpiperidin-4-yl)butyl]-3-phenylprop-2-enamide
Mus musculus
2.4.2.12
gallotanine
i.e. (2R,3S,5R,6S)-tetrahydro-2H-pyran-2,3,4,5,6-pentaylpentakis(oxycarbonyl-5,6-dihydroxybenzene-3,1-diyl) pentakis(3,4,5-trihydroxybenzoate)
Mus musculus
Purification (Commentary) (protein specific)
2.4.2.12
immobilized metal ion affinity chromatography
Mus musculus
Substrates and Products (Substrate) (protein specific)
2.4.2.12
nicotinamide + 5-phosphoribosyl 1-diphosphate
721273
Mus musculus
nicotinamide mononucleotide + diphosphate
?