EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
7.6.2.2 | Diazoxide | about 55% increase in ATPase activity, half-activation concentration is 0.6 mM | Cricetulus griseus | |
7.6.2.2 | glibenclamide | augments the ATPase activity with a maximum attained near 100 microM | Cricetulus griseus | |
7.6.2.2 | meglitinide | increases ATPase activity, maximum activation levels of 70% | Cricetulus griseus | |
7.6.2.2 | additional information | ligands of sulfonylurea receptor SUR also interact with P-plycoprotein, due to structural similarity between drug binding domains in the two proteins | Cricetulus griseus | |
7.6.2.2 | P1075 | about 55% increase in ATPase activity, half-activation concentration is 0.036 mM | Cricetulus griseus | |
7.6.2.2 | SR47063 | 100% increase in ATPase activity, half-activation concentration is 1.5 mM | Cricetulus griseus | |
7.6.2.2 | Tolbutamide | increases ATPase activity, with maximum activation levels of 70% | Cricetulus griseus |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
7.6.2.2 | Cricetulus griseus | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
7.6.2.2 | DC-3F/ADX cell | selected from spontaneously transformed Chinese hamster lung fibroblast DC-3F on the basis of resistance to actinomycin D | Cricetulus griseus | - |