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Literature summary extracted from

  • Koizumi, M.; Momoeda, M.; Hiroi, H.; Nakazawa, F.; Nakae, H.; Ohno, T.; Yano, T.; Taketani, Y.
    Inhibition of proteases involved in embryo implantation by cholesterol sulfate (2010), Hum. Reprod., 25, 192-197.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.21.7 Cholesterol sulfate reduces plasmin activity in a dose-dependent manner Homo sapiens

Organism

EC Number Organism UniProt Comment Textmining
3.4.21.7 Homo sapiens
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.21.7 endometrial stromal cell
-
Homo sapiens
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.21.7 Boc-Val-Leu-Lys-4-methylcoumaryl-7-amide + H2O
-
Homo sapiens Boc-Val-Leu-Lys + 7-amino-4-methylcoumarin
-
?

Synonyms

EC Number Synonyms Comment Organism
3.4.21.7 plasmin
-
Homo sapiens

Temperature Optimum [°C]

EC Number Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
3.4.21.7 37
-
assay at Homo sapiens

pH Optimum

EC Number pH Optimum Minimum pH Optimum Maximum Comment Organism
3.4.21.7 7.5
-
assay at Homo sapiens

General Information

EC Number General Information Comment Organism
3.4.21.7 physiological function Western blot analysis of the endometrial stromal cell culture media reveals that cholesterol sulfate inhibits the conversion by plasmin of matrix metalloproteinase-3 from the precursor form to the active form Homo sapiens