EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
2.7.11.26 | AT7519 | 0.0005 mM AT7519 inhibits glycogen synthase kinase 3beta phosphorylation, AT7519 dephosphorylates GSK-3beta independent of inhibition of transcription | Homo sapiens |
EC Number | Application | Comment | Organism |
---|---|---|---|
2.7.11.26 | medicine | GSK-3beta is a therapeutic target in cancer treatment | Homo sapiens |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.7.11.26 | ATP + beta-catenin | Homo sapiens | - |
ADP + phosphorylated beta-catenin | - |
? | |
2.7.11.26 | ATP + c-Myc | Homo sapiens | - |
ADP + phosphorylated c-Myc | - |
? | |
2.7.11.26 | ATP + cyclin D | Homo sapiens | - |
ADP + phosphorylated cyclin D | - |
? | |
2.7.11.26 | ATP + cyclin E | Homo sapiens | - |
ADP + phosphorylated cyclin E | - |
? | |
2.7.11.26 | ATP + glycogen synthase | Homo sapiens | - |
ADP + glycogen synthase phosphate | - |
? | |
2.7.11.26 | ATP + nuclear factor-kappaB | Homo sapiens | - |
ADP + phosphorylated nuclear factor-kappaB | - |
? | |
2.7.11.26 | ATP + p53 | Homo sapiens | - |
ADP + phosphorylated p53 | - |
? | |
2.7.11.26 | ATP + protein tau | Homo sapiens | - |
ADP + protein tau phosphate | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
2.7.11.26 | Homo sapiens | - |
- |
- |
EC Number | Posttranslational Modification | Comment | Organism |
---|---|---|---|
2.7.11.26 | phosphoprotein | GSK-3beta is activated via phosphorylation at Ser9 | Homo sapiens |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
2.7.11.26 | MM1-S cell | - |
Homo sapiens | - |
2.7.11.26 | multiple myeloma cell | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.7.11.26 | ATP + beta-catenin | - |
Homo sapiens | ADP + phosphorylated beta-catenin | - |
? | |
2.7.11.26 | ATP + c-Myc | - |
Homo sapiens | ADP + phosphorylated c-Myc | - |
? | |
2.7.11.26 | ATP + cyclin D | - |
Homo sapiens | ADP + phosphorylated cyclin D | - |
? | |
2.7.11.26 | ATP + cyclin E | - |
Homo sapiens | ADP + phosphorylated cyclin E | - |
? | |
2.7.11.26 | ATP + glycogen synthase | - |
Homo sapiens | ADP + glycogen synthase phosphate | - |
? | |
2.7.11.26 | ATP + nuclear factor-kappaB | - |
Homo sapiens | ADP + phosphorylated nuclear factor-kappaB | - |
? | |
2.7.11.26 | ATP + p53 | - |
Homo sapiens | ADP + phosphorylated p53 | - |
? | |
2.7.11.26 | ATP + protein tau | - |
Homo sapiens | ADP + protein tau phosphate | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
2.7.11.26 | glycogen synthase kinase-3beta | - |
Homo sapiens |
2.7.11.26 | GSK-3beta | - |
Homo sapiens |
EC Number | Cofactor | Comment | Organism | Structure |
---|---|---|---|---|
2.7.11.26 | ATP | - |
Homo sapiens |