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Literature summary extracted from

  • Fan, C.; Clay, M.D.; Deyholos, M.K.; Vederas, J.C.
    Exploration of inhibitors for diaminopimelate aminotransferase (2010), Bioorg. Med. Chem., 18, 2141-2151.
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
2.6.1.83 expressed in Escherichia coli Arabidopsis thaliana

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.6.1.83 (2-[(E)-[1-(4-chlorophenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)acetic acid 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (2-[(E)-[1-methyl-3-(4-methylphenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)acetic acid 17% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (2E)-2-cyano-3-[5-(dimethylamino)furan-2-yl]-N-(3,4-dimethylphenyl)prop-2-enamide 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (2Z)-N'-nitro-2-[[5-(3-nitrophenyl)furan-2-yl]methylidene]hydrazinecarboximidamide 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (3E)-1-[(4-methoxyphenyl)sulfonyl]-3-[4-oxo-3-(prop-2-en-1-yl)-2-thioxo-1,3-thiazolidin-5-ylidene]-1,3-dihydro-2H-indol-2-one 18% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (3E)-1-[(4-methylphenyl)sulfonyl]-3-(4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)-1,3-dihydro-2H-indol-2-one 25% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (3E)-3-[2-(2,4-dimethyl-1,3-thiazol-5-yl)-2-oxoethylidene]-3,4-dihydroquinoxalin-2(1H)-one 18% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (3E)-3-[2-oxo-2-(thiophen-2-yl)ethylidene]-3,4-dihydroquinoxalin-2(1H)-one 15% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (3Z)-3-(2,4-dimethoxybenzylidene)-5-phenylfuran-2(3H)-one 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5E)-5-(1H-indol-2-ylmethylidene)-1-(4-methylphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 16% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5E)-5-[(1-benzyl-1H-indol-2-yl)methylidene]-1-(2-methoxyphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 20% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5E)-5-[(1-methyl-1H-indol-2-yl)methylidene]-1-(prop-2-en-1-yl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 35% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5E)-5-[(1-methyl-1H-indol-2-yl)methylidene]-1-prop-2-en-1-yl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 45% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5E)-5-[[1-(4-nitrobenzyl)-1H-indol-2-yl]methylidene]-1-(prop-2-en-1-yl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 33% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-1-(3-bromophenyl)-5-(furan-2-ylmethylidene)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 17% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-3-(1,1-dioxidotetrahydrothiophen-3-yl)-5-[[1-phenyl-3-(thiophen-2-yl)-1H-pyrazol-4-yl]methylidene]-2-thioxo-1,3-thiazolidin-4-one 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-(3-iodo-4-methoxybenzylidene)-2-thioxo-1,3-thiazolidin-4-one 29% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[(3-methylthiophen-2-yl)methylidene]-3-(1-phenylethyl)-2-thioxo-1,3-thiazolidin-4-one 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[(3-methylthiophen-2-yl)methylidene]-3-(tetrahydrofuran-2-ylmethyl)-2-thioxo-1,3-thiazolidin-4-one 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[(6-bromo-1,3-benzodioxol-5-yl)methylidene]-2-(4-methylphenyl)-1,3-thiazol-4(5H)-one 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[5-(2-chlorobenzyl)-2-hydroxybenzylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[[5-(2-bromo-4-nitrophenyl)furan-2-yl]methylidene]-2-imino-1,3-thiazolidin-4-one 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (5Z)-5-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-1-(4-methoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione 20% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 (Z)-3-amino-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-3-ethyl-5-(2-hydroxybenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-3-ethyl-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-3-ethyl-5-(naphthalen-1-ylmethylene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-3-ethyl-5-(quinolin-5-ylmethylene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-(2-hydroxybenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-(4-(dimethylamino)benzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-(4-chlorobenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-(4-chlorobenzylidene)-3-ethyl-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-5-benzylidene-3-ethyl-2-thioxothiazolidin-4-one
-
 Arabidopsis thaliana
2.6.1.83 (Z)-N -(5-((5-(4-nitrophenyl)furan-2-yl)methylene)-4-oxo-2-thioxothiazolidin-3-yl)acetamide
-
 Arabidopsis thaliana
2.6.1.83 (Z)-N-(5-(4-methoxybenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetamide
-
 Arabidopsis thaliana
2.6.1.83 1,3-dimethyl-5-[[1-(3-nitrophenyl)-1H-pyrrol-2-yl]methylidene]pyrimidine-2,4,6(1H,3H,5H)-trione 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 1-(4-fluorophenyl)-2-[[4-phenyl-5-(3,4,5-trimethoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]ethanone 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 2-(2-[(E)-[1-(4-fluorophenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)-N-phenylacetamide 18% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 2-thioxo-5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylidene]dihydropyrimidine-4,6(1H,5H)-dione 15% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 2-[(2E)-2-(2-oxo-5-phenylfuran-3(2H)-ylidene)hydrazinyl]benzoic acid 16% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 3-cyclopropyl-N'-[(1E)-1-(4-methylphenyl)ethylidene]-1H-pyrazole-5-carbohydrazide 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 3-[2-[(4-acetylphenyl)amino]-1,3-thiazol-4-yl]-2H-chromen-2-one 16% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 4-[(E)-[2-(2-chlorophenyl)-5-oxo-1,3-oxazol-4(5H)-ylidene]methyl]-2-hydroxyphenyl 2-chlorobenzoate 30% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 5-(4-methylphenyl)-4-[[(E)-(2,4,5-trimethoxyphenyl)methylidene]amino]-4H-1,2,4-triazole-3-thiol 18% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 5-([1-[2-(3,4-dimethylphenoxy)ethyl]-1H-indol-2-yl]methylidene)pyrimidine-2,4,6(1H,3H,5H)-trione 28% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 5-[(5-hydroxy-1-phenyl-1H-pyrazol-4-yl)methylidene]-1,3-dimethylpyrimidine-2,4,6(1H,3H,5H)-trione 20% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 5-[3-[(2-chlorobenzyl)oxy]-4-methoxybenzylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 48% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 8-methoxy-3-[(2-methylprop-2-en-1-yl)oxy]-6H-benzo[c]chromen-6-one 25% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 ethyl (5Z)-5-[[4-(dimethylamino)phenyl]methylidene]-2-[(4-methoxyphenyl)amino]-4-oxo-4,5-dihydrothiophene-3-carboxylate 22% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 ethyl (5Z)-5-[[4-(dimethylamino)phenyl]methylidene]-2-[(4-nitrophenyl)amino]-4-oxo-4,5-dihydrothiophene-3-carboxylate 19% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 ethyl 4-(5-[(Z)-[2,4,6-trioxo-1-(prop-2-en-1-yl)tetrahydropyrimidin-5(2H)-ylidene]methyl]furan-2-yl)benzoate 16% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 additional information not inhibited by (Z)-5-benzylidene-2-thioxothiazolidin-4-one, (Z)-5-(naphthalen-1-ylmethylene)-2-thioxothiazolidin-4-one, (Z)-3-amino-5-benzylidene-2-thioxothiazolidin-4-one, (Z)-3-amino-5-(4-chlorobenzylidene)-2-thioxothiazolidin-4-one, (Z)-N-(5-benzylidene-4-oxo-2-thioxothiazolidin-3-yl)-acetamide, (Z)-N-(5-(4-chlorobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetamide, and (Z)-5-(2-nitrobenzylidene)-2-thioxothiazolidin-4-one Arabidopsis thaliana
2.6.1.83 N'-[(E)-(2,4-dihydroxyphenyl)methylidene]-5-nitro-3-phenyl-1H-indole-2-carbohydrazide 15% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N'-[(Z)-(4-fluorophenyl)methylidene]-3-(naphthalen-2-yl)-1H-pyrazole-5-carbohydrazide 14% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N-[(2E,5Z)-5-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetamide 52% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N-[(5E)-5-[(5-bromofuran-2-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetamide 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N-[3-(hydrazinylcarbonyl)naphthalen-2-yl]benzenesulfonamide 33% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N-[3-[(2,5-dimethoxyphenyl)amino]quinoxalin-2-yl]-3-nitrobenzenesulfonamide 13% inhibition at 0.01 mM Arabidopsis thaliana
2.6.1.83 N-[[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]carbamothioyl]-3-methyl-1-benzofuran-2-carboxamide 19% inhibition at 0.01 mM Arabidopsis thaliana

Organism

EC Number Organism UniProt Comment Textmining
2.6.1.83 Arabidopsis thaliana
-
-
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2.6.1.83 L-2-amino-6-oxopimelate + L-glutamate + H2O
-
 Arabidopsis thaliana LL-2,6-diaminopimelate + 2-oxoglutarate
-
 ?

Synonyms

EC Number Synonyms Comment Organism
2.6.1.83 diaminopimelate aminotransferase
-
 Arabidopsis thaliana
2.6.1.83 LL-DAP-AT
-
 Arabidopsis thaliana

Cofactor

EC Number Cofactor Comment Organism Structure
2.6.1.83 pyridoxal 5'-phosphate
-
 Arabidopsis thaliana

IC50 Value

EC Number IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
2.6.1.83 0.005
-
-
 Arabidopsis thaliana N-[3-(hydrazinylcarbonyl)naphthalen-2-yl]benzenesulfonamide
2.6.1.83 0.025
-
-
 Arabidopsis thaliana 2-thioxo-5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylidene]dihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.031
-
-
 Arabidopsis thaliana (3E)-3-[2-oxo-2-(thiophen-2-yl)ethylidene]-3,4-dihydroquinoxalin-2(1H)-one
2.6.1.83 0.033
-
-
 Arabidopsis thaliana (5E)-5-[(1-methyl-1H-indol-2-yl)methylidene]-1-prop-2-en-1-yl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.037
-
-
 Arabidopsis thaliana (2-[(E)-[1-methyl-3-(4-methylphenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)acetic acid
2.6.1.83 0.039
-
-
 Arabidopsis thaliana 2-[(2E)-2-(2-oxo-5-phenylfuran-3(2H)-ylidene)hydrazinyl]benzoic acid
2.6.1.83 0.041
-
-
 Arabidopsis thaliana N-[(5E)-5-[(5-bromofuran-2-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetamide
2.6.1.83 0.042
-
-
 Arabidopsis thaliana (5Z)-5-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-1-(4-methoxyphenyl)pyrimidine-2,4,6(1H,3H,5H)-trione
2.6.1.83 0.045
-
-
 Arabidopsis thaliana 5-[(5-hydroxy-1-phenyl-1H-pyrazol-4-yl)methylidene]-1,3-dimethylpyrimidine-2,4,6(1H,3H,5H)-trione
2.6.1.83 0.045
-
-
 Arabidopsis thaliana N'-[(E)-(2,4-dihydroxyphenyl)methylidene]-5-nitro-3-phenyl-1H-indole-2-carbohydrazide
2.6.1.83 0.046
-
-
 Arabidopsis thaliana (5Z)-5-[5-(2-chlorobenzyl)-2-hydroxybenzylidene]-3-ethyl-2-thioxo-1,3-thiazolidin-4-one
2.6.1.83 0.052
-
-
 Arabidopsis thaliana 2-(2-[(E)-[1-(4-fluorophenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)-N-phenylacetamide
2.6.1.83 0.056
-
-
 Arabidopsis thaliana (3E)-3-[2-(2,4-dimethyl-1,3-thiazol-5-yl)-2-oxoethylidene]-3,4-dihydroquinoxalin-2(1H)-one
2.6.1.83 0.062
-
-
 Arabidopsis thaliana (5E)-5-[(1-benzyl-1H-indol-2-yl)methylidene]-1-(2-methoxyphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.065
-
-
 Arabidopsis thaliana (2-[(E)-[1-(4-chlorophenyl)-2,4,6-trioxotetrahydropyrimidin-5(2H)-ylidene]methyl]-1H-indol-1-yl)acetic acid
2.6.1.83 0.069
-
-
 Arabidopsis thaliana (5E)-5-[[1-(4-nitrobenzyl)-1H-indol-2-yl]methylidene]-1-(prop-2-en-1-yl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.07
-
-
 Arabidopsis thaliana (3E)-1-[(4-methylphenyl)sulfonyl]-3-(4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)-1,3-dihydro-2H-indol-2-one
2.6.1.83 0.073
-
 in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-N -(5-((5-(4-nitrophenyl)furan-2-yl)methylene)-4-oxo-2-thioxothiazolidin-3-yl)acetamide
2.6.1.83 0.075
-
-
 Arabidopsis thaliana (5E)-5-[(1-methyl-1H-indol-2-yl)methylidene]-1-(prop-2-en-1-yl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.078
-
-
 Arabidopsis thaliana N-[(2E,5Z)-5-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetamide
2.6.1.83 0.081
-
-
 Arabidopsis thaliana 4-[(E)-[2-(2-chlorophenyl)-5-oxo-1,3-oxazol-4(5H)-ylidene]methyl]-2-hydroxyphenyl 2-chlorobenzoate
2.6.1.83 0.083
-
-
 Arabidopsis thaliana N-[[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]carbamothioyl]-3-methyl-1-benzofuran-2-carboxamide
2.6.1.83 0.085
-
-
 Arabidopsis thaliana (5Z)-5-[[5-(2-bromo-4-nitrophenyl)furan-2-yl]methylidene]-2-imino-1,3-thiazolidin-4-one
2.6.1.83 0.099
-
-
 Arabidopsis thaliana 5-([1-[2-(3,4-dimethylphenoxy)ethyl]-1H-indol-2-yl]methylidene)pyrimidine-2,4,6(1H,3H,5H)-trione
2.6.1.83 0.117
-
-
 Arabidopsis thaliana (5Z)-3-(1,1-dioxidotetrahydrothiophen-3-yl)-5-[[1-phenyl-3-(thiophen-2-yl)-1H-pyrazol-4-yl]methylidene]-2-thioxo-1,3-thiazolidin-4-one
2.6.1.83 0.121
-
-
 Arabidopsis thaliana 5-[3-[(2-chlorobenzyl)oxy]-4-methoxybenzylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.127
-
-
 Arabidopsis thaliana (5Z)-5-[(3-methylthiophen-2-yl)methylidene]-3-(1-phenylethyl)-2-thioxo-1,3-thiazolidin-4-one
2.6.1.83 0.127
-
 in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-(4-(dimethylamino)benzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.13
-
-
 Arabidopsis thaliana (5Z)-5-[(6-bromo-1,3-benzodioxol-5-yl)methylidene]-2-(4-methylphenyl)-1,3-thiazol-4(5H)-one
2.6.1.83 0.141
-
-
 Arabidopsis thaliana ethyl (5Z)-5-[[4-(dimethylamino)phenyl]methylidene]-2-[(4-nitrophenyl)amino]-4-oxo-4,5-dihydrothiophene-3-carboxylate
2.6.1.83 0.142
-
 in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.153
-
-
 Arabidopsis thaliana N-[3-[(2,5-dimethoxyphenyl)amino]quinoxalin-2-yl]-3-nitrobenzenesulfonamide
2.6.1.83 0.155
-
 in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-3-amino-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.159
-
-
 Arabidopsis thaliana (3Z)-3-(2,4-dimethoxybenzylidene)-5-phenylfuran-2(3H)-one
2.6.1.83 0.161
-
-
 Arabidopsis thaliana N'-[(Z)-(4-fluorophenyl)methylidene]-3-(naphthalen-2-yl)-1H-pyrazole-5-carbohydrazide
2.6.1.83 0.164
-
-
 Arabidopsis thaliana (5E)-5-(1H-indol-2-ylmethylidene)-1-(4-methylphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.18
-
-
 Arabidopsis thaliana (5Z)-5-(3-iodo-4-methoxybenzylidene)-2-thioxo-1,3-thiazolidin-4-one
2.6.1.83 0.19
-
 in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-3-ethyl-5-(quinolin-5-ylmethylene)-2-thioxothiazolidin-4-one
2.6.1.83 0.194
-
-
 Arabidopsis thaliana (3E)-1-[(4-methoxyphenyl)sulfonyl]-3-[4-oxo-3-(prop-2-en-1-yl)-2-thioxo-1,3-thiazolidin-5-ylidene]-1,3-dihydro-2H-indol-2-one
2.6.1.83 0.2
-
-
 Arabidopsis thaliana (5Z)-1-(3-bromophenyl)-5-(furan-2-ylmethylidene)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana ethyl (5Z)-5-[[4-(dimethylamino)phenyl]methylidene]-2-[(4-methoxyphenyl)amino]-4-oxo-4,5-dihydrothiophene-3-carboxylate
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana (5Z)-5-[(3-methylthiophen-2-yl)methylidene]-3-(tetrahydrofuran-2-ylmethyl)-2-thioxo-1,3-thiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana ethyl 4-(5-[(Z)-[2,4,6-trioxo-1-(prop-2-en-1-yl)tetrahydropyrimidin-5(2H)-ylidene]methyl]furan-2-yl)benzoate
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 1,3-dimethyl-5-[[1-(3-nitrophenyl)-1H-pyrrol-2-yl]methylidene]pyrimidine-2,4,6(1H,3H,5H)-trione
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana (2E)-2-cyano-3-[5-(dimethylamino)furan-2-yl]-N-(3,4-dimethylphenyl)prop-2-enamide
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 3-cyclopropyl-N'-[(1E)-1-(4-methylphenyl)ethylidene]-1H-pyrazole-5-carbohydrazide
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana (2Z)-N'-nitro-2-[[5-(3-nitrophenyl)furan-2-yl]methylidene]hydrazinecarboximidamide
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 3-[2-[(4-acetylphenyl)amino]-1,3-thiazol-4-yl]-2H-chromen-2-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 8-methoxy-3-[(2-methylprop-2-en-1-yl)oxy]-6H-benzo[c]chromen-6-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 5-(4-methylphenyl)-4-[[(E)-(2,4,5-trimethoxyphenyl)methylidene]amino]-4H-1,2,4-triazole-3-thiol
2.6.1.83 0.2
-
 IC50 above 0.2 mM Arabidopsis thaliana 1-(4-fluorophenyl)-2-[[4-phenyl-5-(3,4,5-trimethoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl]ethanone
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-(4-chlorobenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-(2-hydroxybenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-benzylidene-3-ethyl-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-3-ethyl-5-(2-hydroxybenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-3-ethyl-5-(4-methoxybenzylidene)-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-5-(4-chlorobenzylidene)-3-ethyl-2-thioxothiazolidin-4-one
2.6.1.83 0.2
-
 IC50 above 0.2 mM, in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-N-(5-(4-methoxybenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetamide
2.6.1.83 0.2
-
 IC50 above 0.2 mM,in 100 mM HEPES-KOH, pH 7.6 Arabidopsis thaliana (Z)-3-ethyl-5-(naphthalen-1-ylmethylene)-2-thioxothiazolidin-4-one