EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.14.5 | saxagliptin | highly potent and selective inhibitor of DPP-IV | Homo sapiens | |
3.4.14.5 | sitagliptin | selective inhibitor of DPP-IV, over 80% inhibition of DPP-IV with a single oral dose of 50 mg | Homo sapiens | |
3.4.14.5 | vildagliptin | highly potent and stable selective inhibitor of DPP-IV, over 90% inhibition of DPP-IV with a single oral dose of 100 mg | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.14.5 | Homo sapiens | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.14.5 | breast | - |
Homo sapiens | - |
3.4.14.5 | endothelial cell | - |
Homo sapiens | - |
3.4.14.5 | intestine | - |
Homo sapiens | - |
3.4.14.5 | kidney | most densely located in the kidney | Homo sapiens | - |
3.4.14.5 | liver | - |
Homo sapiens | - |
3.4.14.5 | lymphocyte | - |
Homo sapiens | - |
3.4.14.5 | macrophage | - |
Homo sapiens | - |
3.4.14.5 | ovary | - |
Homo sapiens | - |
3.4.14.5 | placenta | - |
Homo sapiens | - |
3.4.14.5 | thyroid gland | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.14.5 | glucagon-like peptide 1 + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | glucose-dependent insulinotropic peptide + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | growth hormone-releasing hormone + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | neuropeptide Y + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | peptide YY + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | pituitary adenylate cyclase activating peptide + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.14.5 | Substance P + H2O | - |
Homo sapiens | ? | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.14.5 | dipeptidyl peptidase-IV | - |
Homo sapiens |
3.4.14.5 | DPP-IV | - |
Homo sapiens |