EC Number | Crystallization (Comment) | Organism |
---|---|---|
6.5.1.3 | virtual screen of REL1 crystal structure for inhibitors | Trypanosoma brucei |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
6.5.1.3 | 1-amino-4-(3-(aminosulfonyl)anilino)-9,10-dioxo-9,10-dihydro-2-anthracenesulfonic acid | 68.5% residual activity at 0.01 mM, presence of Triton X-100. Molecular dynamics simulations | Trypanosoma brucei | |
6.5.1.3 | 3-((4-(ethylamino)phenyl)diazenyl)-4,5-dihydroxy-2,7-naphthalenedisulfonic acid | 4.1% residual activity at 0.01 mM, presence of Triton X-100. Molecular dynamics simulations | Trypanosoma brucei | |
6.5.1.3 | 3-((5-chloro-2-hydroxyphenyl)diazenyl)-4,5-dihydroxy-2,7-naphthalenedisulfonic acid | 8.6% residual activity at 0.01 mM, presence of Triton X-100. Molecular dynamics simulations | Trypanosoma brucei | |
6.5.1.3 | 4,5-dihydroxy-3-(1-naphthyldiazenyl)-2,7-naphthalenedisulfonic acid | 43.1% residual activity at 0.01 mM, presence of Triton X-100. Molecular dynamics simulations | Trypanosoma brucei |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
6.5.1.3 | Trypanosoma brucei | P86927 | - |
- |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
6.5.1.3 | REL1 | - |
Trypanosoma brucei |
6.5.1.3 | RNA-editing ligase 1 | - |
Trypanosoma brucei |