Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary extracted from

  • Dai, R.; Ali, M.K.; Lezcano, N.; Bergson, C.
    A crucial role for cAMP and protein kinase A in D1 dopamine receptor regulated intracellular calcium transients (2008), Neurosignals, 16, 112-123.
    View publication on PubMed

Activating Compound

EC Number Activating Compound Comment Organism Structure
2.7.11.11 8-bromo-cAMP 1 mM Homo sapiens
2.7.11.11 8-bromo-cAMP 1 mM Rattus norvegicus
2.7.11.11 forskolin 0.01 mM Homo sapiens
2.7.11.11 forskolin 0.01 mM Rattus norvegicus

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.11.11 H-89
-
Homo sapiens
2.7.11.11 H-89
-
Rattus norvegicus
2.7.11.11 KT-5720
-
Homo sapiens
2.7.11.11 KT-5720
-
Rattus norvegicus

Organism

EC Number Organism UniProt Comment Textmining
2.7.11.11 Homo sapiens
-
-
-
2.7.11.11 Rattus norvegicus
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
2.7.11.11 D1-HEK-293 cell HEK-293 cells that stably express D1 receptors Homo sapiens
-
2.7.11.11 hippocampus
-
Rattus norvegicus
-
2.7.11.11 neuron
-
Rattus norvegicus
-

Synonyms

EC Number Synonyms Comment Organism
2.7.11.11 PKA
-
Homo sapiens
2.7.11.11 PKA
-
Rattus norvegicus
2.7.11.11 protein kinase A
-
Homo sapiens
2.7.11.11 protein kinase A
-
Rattus norvegicus

Cofactor

EC Number Cofactor Comment Organism Structure
2.7.11.11 ATP
-
Homo sapiens
2.7.11.11 ATP
-
Rattus norvegicus
2.7.11.11 cAMP dependent Homo sapiens
2.7.11.11 cAMP dependent Rattus norvegicus