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Literature summary extracted from

  • De Arcangelis, V.; Soto, D.; Xiang, Y.
    Phosphodiesterase 4 and phosphatase 2A differentially regulate cAMP/protein kinase a signaling for cardiac myocyte contraction under stimulation of beta1 adrenergic receptor (2008), Mol. Pharmacol., 74, 1453-1462.
    View publication on PubMedView publication on EuropePMC

Activating Compound

EC Number Activating Compound Comment Organism Structure
3.1.4.53 isoproterenol PDE4 activity is stimulated with 0.01 mM isoproterenol Mus musculus

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.4.53 rolipram
-
Mus musculus

Organism

EC Number Organism UniProt Comment Textmining
3.1.4.53 Mus musculus
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.4.53 cardiac myocyte
-
Mus musculus
-
3.1.4.53 heart
-
Mus musculus
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.1.4.53 3',5'-cAMP + H2O
-
Mus musculus 5'-AMP
-
?

Synonyms

EC Number Synonyms Comment Organism
3.1.4.53 PDE4
-
Mus musculus
3.1.4.53 phosphodiesterase 4
-
Mus musculus