EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
4.6.1.1 | A-77636 | a dopamine receptor agonist, the activation by can be reversed by D1-receptor antagonists SCH23390, SKF83566, and butaclamol | Rattus norvegicus | |
4.6.1.1 | dihydrexidine | a dopamine receptor agonist, the activation by can be reversed by D1-receptor antagonists SCH23390, SKF83566, and butaclamol | Rattus norvegicus | |
4.6.1.1 | dopamine | a dopamine receptor agonist, the activation by can be reversed by D1-receptor antagonists SCH23390, SKF83566, and butaclamol | Rattus norvegicus | |
4.6.1.1 | forskolin | activation in a Mg2+-dependent manner | Rattus norvegicus | |
4.6.1.1 | additional information | measurement of dopamine receptor agonist activation in a competitive assay with antagonists, e.g. SCH23390, overview | Rattus norvegicus |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
4.6.1.1 | Mg2+ | Mg2+ is required for forskolin-dependent accumulation of cAMP, best at 1-3 mM | Rattus norvegicus |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
4.6.1.1 | ATP | Rattus norvegicus | - |
3',5'-cyclic-AMP + diphosphate | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
4.6.1.1 | Rattus norvegicus | - |
Wistar rats | - |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
4.6.1.1 | brain | - |
Rattus norvegicus | - |
4.6.1.1 | striatum | - |
Rattus norvegicus | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
4.6.1.1 | ATP | - |
Rattus norvegicus | 3',5'-cyclic-AMP + diphosphate | - |
? |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
4.6.1.1 | 30 | - |
assay at | Rattus norvegicus |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
4.6.1.1 | 7.4 | - |
assay at | Rattus norvegicus |