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Literature summary extracted from

  • Taylor, S.S.; Kim, C.; Cheng, C.Y.; Brown, S.H.; Wu, J.; Kannan, N.
    Signaling through cAMP and cAMP-dependent protein kinase: diverse strategies for drug design (2008), Biochim. Biophys. Acta, 1784, 16-26.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.11.11 PKA regulatory subunit Ialpha pseudosubstrate inhibitor Homo sapiens
2.7.11.11 PKI pseudosubstrate inhibitor Homo sapiens
2.7.11.11 RIIalpha subunit
-
Homo sapiens

Organism

EC Number Organism UniProt Comment Textmining
2.7.11.11 Homo sapiens
-
-
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2.7.11.11 ATP + PKA regulatory subunit IIalpha
-
Homo sapiens ADP + phosphorylated PKA regulatory subunit IIalpha
-
?

Synonyms

EC Number Synonyms Comment Organism
2.7.11.11 PKA
-
Homo sapiens

Cofactor

EC Number Cofactor Comment Organism Structure
2.7.11.11 ATP
-
Homo sapiens
2.7.11.11 cAMP dependent Homo sapiens