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Literature summary extracted from

  • Moro, C.; Klimcakova, E.; Lafontan, M.; Berlan, M.; Galitzky, J.
    Phosphodiesterase-5A and neutral endopeptidase activities in human adipocytes do not control atrial natriuretic peptide-mediated lipolysis (2007), Br. J. Pharmacol., 152, 1102-1110.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.24.11 thiorphan
-
Homo sapiens

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.4.24.11 membrane
-
Homo sapiens 16020
-

Molecular Weight [Da]

EC Number Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
3.4.24.11 94000
-
-
Homo sapiens

Organism

EC Number Organism UniProt Comment Textmining
3.4.24.11 Homo sapiens
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.24.11 adipocyte adipocyte membrane Homo sapiens
-

Specific Activity [micromol/min/mg]

EC Number Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
3.4.24.11 0.0000018
-
on human adipocyte membranes Homo sapiens

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.4.24.11 0.00191
-
thiorphan
-
Homo sapiens