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Literature summary extracted from

  • Wu, J.J.; Fujikawa, K.; McMullen, B.A.; Chung, D.W.
    Characterization of a core binding site for ADAMTS-13 in the A2 domain of von Willebrand factor (2006), Proc. Natl. Acad. Sci. USA, 103, 18470-18474.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.24.87 Pro-1645-Lys-1668 fragment of von Willebrand factor 73
-
Homo sapiens

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.24.87 0.00025
-
HRPH-A2-B
-
Homo sapiens

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.4.24.87 von Willebrand factor + H2O Homo sapiens
-
?
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.4.24.87 Homo sapiens
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.24.87 blood plasma
-
Homo sapiens
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.24.87 HRPH-A2-B HRPH-A2-B is a derivative of von Willebrand factor 73, consisting of a HRP conjugate of a biotinylated von Willebrand factor 78 sequence Homo sapiens ? cleavage of Tyr842-Met843 within the A2 domain, i.e. Tyr1605-Met1606 in von Willebrand factor UniProt Id P04275 ?
3.4.24.87 von Willebrand factor + H2O
-
Homo sapiens ?
-
?
3.4.24.87 von Willebrand factor 73 + H2O minimal substrate cleavable by ADAMTS-13 Homo sapiens ?
-
?

Synonyms

EC Number Synonyms Comment Organism
3.4.24.87 ADAMTS-13
-
Homo sapiens

Turnover Number [1/s]

EC Number Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
3.4.24.87 0.67
-
HRPH-A2-B
-
Homo sapiens

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.4.24.87 0.012
-
Pro-1645-Lys-1668 fragment of von Willebrand factor 73
-
Homo sapiens