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Literature summary extracted from

  • Levesque, S.A.; Lavoie, E.G.; Lecka, J.; Bigonnesse, F.; Sevigny, J.
    Specificity of the ecto-ATPase inhibitor ARL 67156 on human and mouse ectonucleotidases (2007), Br. J. Pharmacol., 152, 141-150.
    View publication on PubMedView publication on EuropePMC

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.3.5 6-N,N-diethyl-D-beta-gamma-dibromomethylene adenosine triphosphate originally named FPL 67156 or ARL 67156, 28% inhibition at 0.1 mM Homo sapiens
3.1.3.5 ADP 40% inhibition at 0.1 mM Homo sapiens
3.1.3.5 alpha,beta-methylene-ADP highly effective competitive inhibitor Homo sapiens
3.1.3.5 ATP 70% inhibition at 0.1 mM Homo sapiens

Organism

EC Number Organism UniProt Comment Textmining
3.1.3.5 Homo sapiens Q53Z63
-
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.1.3.5 5'-AMP + H2O
-
 Homo sapiens adenosine + phosphate
-
 ?

Synonyms

EC Number Synonyms Comment Organism
3.1.3.5 ecto-5'-nucleotidase
-
 Homo sapiens
3.1.3.5 ectonucleotidase
-
 Homo sapiens