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Literature summary extracted from

  • Chiou, S.Y.; Lai, G.W.; Tsai, Y.H.; Lee, Y.R.; Lin, L.Y.; Lin, G.L.
    Kinetics and mechanisms of acetylcholinesterase and butyrylcholinesterase inhibition by cardiovascular drugs and benzodiazepines (2005), J. Chin. Chem. Soc., 52, 843-848.
No PubMed abstract available

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.1.7 amlodipine besylate
-
Electrophorus electricus
3.1.1.7 chlordiazepoxide HCl
-
Electrophorus electricus
3.1.1.7 diazepam
-
Electrophorus electricus
3.1.1.7 hydralazine HCl
-
Electrophorus electricus
3.1.1.7 lovastatin
-
Electrophorus electricus
3.1.1.7 nifedipine
-
Electrophorus electricus
3.1.1.7 simvastatin
-
Electrophorus electricus
3.1.1.8 amlodipine besylate
-
Equus caballus
3.1.1.8 chlordiazepoxide HCl
-
Equus caballus
3.1.1.8 diazepam
-
Equus caballus
3.1.1.8 hydralazine HCl
-
Equus caballus
3.1.1.8 lovastatin
-
Equus caballus
3.1.1.8 nifedipine
-
Equus caballus
3.1.1.8 simvastatin
-
Equus caballus

Organism

EC Number Organism UniProt Comment Textmining
3.1.1.7 Electrophorus electricus
-
-
-
3.1.1.8 Equus caballus
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.1.8 serum
-
Equus caballus
-

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.1.1.7 0.00019
-
amlodipine besylate
-
Electrophorus electricus
3.1.1.7 0.0018
-
simvastatin
-
Electrophorus electricus
3.1.1.7 0.0027
-
lovastatin
-
Electrophorus electricus
3.1.1.7 0.004
-
nifedipine
-
Electrophorus electricus
3.1.1.7 0.007
-
hydralazine HCl
-
Electrophorus electricus
3.1.1.7 0.013
-
diazepam
-
Electrophorus electricus
3.1.1.7 0.05
-
chlordiazepoxide HCl
-
Electrophorus electricus
3.1.1.8 0.000043
-
diazepam
-
Equus caballus
3.1.1.8 0.00011
-
amlodipine besylate
-
Equus caballus
3.1.1.8 0.0003
-
chlordiazepoxide HCl
-
Equus caballus
3.1.1.8 0.00075
-
simvastatin
-
Equus caballus
3.1.1.8 0.0011
-
lovastatin
-
Equus caballus
3.1.1.8 0.0012
-
nifedipine
-
Equus caballus
3.1.1.8 0.0019
-
hydralazine HCl
-
Equus caballus