EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.21.68 | 2,7-bis-(4-amidinobenzylidene)-cycloheptanone-(1)dihydrochloride | - |
Mus musculus | |
3.4.21.68 | 2,7-bis-(4-amidinobenzylidene)-cycloheptanone-(1)dihydrochloride | - |
Rattus norvegicus |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.21.68 | plasminogen + H2O | Mus musculus | - |
plasmin + ? | - |
? | |
3.4.21.68 | plasminogen + H2O | Rattus norvegicus | - |
plasmin + ? | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.21.68 | Mus musculus | P11214 | - |
- |
3.4.21.68 | Rattus norvegicus | P19637 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.21.68 | brain | primary hippocampal neuron | Mus musculus | - |
3.4.21.68 | brain | primary hippocampal neuron | Rattus norvegicus | - |
3.4.21.68 | Neuro-2a cell | - |
Mus musculus | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.21.68 | plasminogen + H2O | - |
Mus musculus | plasmin + ? | - |
? | |
3.4.21.68 | plasminogen + H2O | - |
Rattus norvegicus | plasmin + ? | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.21.68 | Tissue plasminogen activator | - |
Mus musculus |
3.4.21.68 | Tissue plasminogen activator | - |
Rattus norvegicus |
3.4.21.68 | tPA | - |
Mus musculus |
3.4.21.68 | tPA | - |
Rattus norvegicus |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.21.68 | 0.000035 | - |
2,7-bis-(4-amidinobenzylidene)-cycloheptanone-(1)dihydrochloride | - |
Mus musculus | |
3.4.21.68 | 0.000035 | - |
2,7-bis-(4-amidinobenzylidene)-cycloheptanone-(1)dihydrochloride | - |
Rattus norvegicus |