Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary extracted from

  • Shariat-Madar, Z.; Mahdi, F.; Schmaier, A.H.
    Recombinant prolylcarboxypeptidase activates plasma prekallikrein (2004), Blood, 103, 4554-4561.
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
3.4.16.2 cloned in pMT/BIP/V5-HIS-C, transfected into Scheider insect cells Homo sapiens

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.16.2 angiotensin II
-
Homo sapiens
3.4.16.2 bradykinin
-
Homo sapiens
3.4.16.2 diisopropyl fluorophosphonate
-
Homo sapiens
3.4.16.2 leupeptin
-
Homo sapiens
3.4.16.2 additional information no inhibition by 1 mM EDTA, bradykinin1-5, or angiotensin 1-7 Homo sapiens
3.4.16.2 phenylmethylsulfonyl fluoride
-
Homo sapiens
3.4.16.2 Z-Pro-prolinal
-
Homo sapiens

Metals/Ions

EC Number Metals/Ions Comment Organism Structure
3.4.16.2 Ca2+ optimal activity at 0.01 mM Ca2+ and 1 mM Mg2+ Homo sapiens
3.4.16.2 Mg2+ optimal activity at 0.01 mM Ca2+ and 1 mM Mg2+ Homo sapiens

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3.4.16.2 additional information Homo sapiens the enzyme is a plasma prekallikrein activator ?
-
?

Organism

EC Number Organism UniProt Comment Textmining
3.4.16.2 Homo sapiens
-
-
-

Purification (Commentary)

EC Number Purification (Comment) Organism
3.4.16.2 recombinant Homo sapiens

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.16.2 HUVEC cell
-
Homo sapiens
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.16.2 additional information the enzyme is a plasma prekallikrein activator Homo sapiens ?
-
?

pH Optimum

EC Number pH Optimum Minimum pH Optimum Maximum Comment Organism
3.4.16.2 7.1
-
-
Homo sapiens