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Literature summary extracted from

  • Coimbra, E.S.; Goncalves-da-Costa, S.C.; Corte-Real, S.; De Freitas, F.G.; Durao, A.C.; Souza, C.S.; Silva-Santos, M.I.; Vasconcelos, E.G.
    Characterization and cytochemical localization of an ATP diphosphohydrolase from Leishmania amazonensis promastigotes (2002), Parasitology, 124, 137-143.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.6.1.5 additional information not inhibitory: vanadate, ouabain, thapsigargin, dicyclohexylcarbodiimide, oligomycin, bafilomycin A, levamisole, ammonium molybdate Leishmania amazonensis
3.6.1.5 Sodium azide
-
Leishmania amazonensis

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.6.1.5 plasma membrane
-
Leishmania amazonensis 5886
-

Metals/Ions

EC Number Metals/Ions Comment Organism Structure
3.6.1.5 Ca2+ best activating kation Leishmania amazonensis
3.6.1.5 Co2+ at 1 mM, 73% of ATPase activity compared to Ca2+ Leishmania amazonensis
3.6.1.5 Mg2+ at 1 mM, 61% of ATPase activity compared to Ca2+ Leishmania amazonensis
3.6.1.5 Mn2+ at 1 mM, 65% of ATPase activity compared to Ca2+ Leishmania amazonensis
3.6.1.5 Zn2+ at 1 mM, 70% of ATPase activity compared to Ca2+ Leishmania amazonensis

Organism

EC Number Organism UniProt Comment Textmining
3.6.1.5 Leishmania amazonensis
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.6.1.5 promastigote surface and flagellar pocket Leishmania amazonensis
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.6.1.5 5'-AMP + H2O 23% of activity compared to ATP Leishmania amazonensis adenosine + phosphate
-
?
3.6.1.5 ADP + H2O 104% of activity compared to ATP Leishmania amazonensis AMP + phosphate
-
?
3.6.1.5 ATP + 2 H2O
-
Leishmania amazonensis AMP + 2 phosphate
-
?
3.6.1.5 CTP + 2 H2O 60% of activity compared to ATP Leishmania amazonensis CMP + 2 phosphate
-
?
3.6.1.5 GTP + 2 H2O 23% of activity compared to ATP Leishmania amazonensis GMP + 2 phosphate
-
?
3.6.1.5 UTP + 2 H2O 150% of activity compared to ATP Leishmania amazonensis UMP + 2 phosphate
-
?