Literature summary extracted from
Okafor, C.; Liao, R.; Perreault-Micale, C.; Li, X.; Ito, T.; Stepanek, A.; Doye, A.; de Tombe, P.; Gwathmey, J.K.
Mg-ATPase and Ca+ activated myosin AtPase activity in ventricular myofibrils from non-failing and diseased human hearts--effects of calcium sensitizing agents MCI-154, DPI 201-106, and caffeine (2003), Mol. Cell. Biochem., 245, 77-89.
Activating Compound
EC Number |
Activating Compound |
Comment |
Organism |
Structure |
---|
5.6.1.8 |
Caffeine |
increase in enzyme activity by 4% for non-failing, 11% for idiopathic and 10% ischemic cardiomyopathic hearts |
Homo sapiens |
|
5.6.1.8 |
DPI201-206 |
increase in enzyme activity by less than 5% for all preparations |
Homo sapiens |
|
5.6.1.8 |
MCI-154 |
increase in enzyme activity by 11% for non-failing, 19% for idiopathic and 24% ischemic cardiomyopathic hearts |
Homo sapiens |
|
Application
EC Number |
Application |
Comment |
Organism |
---|
5.6.1.8 |
medicine |
decrease of enzyme activity in hearts of idiopathic and ischemic cardiomyopathic individuals, MCI-154 and caffeine increased enzyme activity |
Homo sapiens |
Localization
EC Number |
Localization |
Comment |
Organism |
GeneOntology No. |
Textmining |
---|
Organism
EC Number |
Organism |
UniProt |
Comment |
Textmining |
---|
5.6.1.8 |
Homo sapiens |
- |
non-failing, idiopathic and ischemic cardiomyopathic individuals |
- |
Source Tissue
EC Number |
Source Tissue |
Comment |
Organism |
Textmining |
---|
5.6.1.8 |
heart |
left ventricular myofibril |
Homo sapiens |
- |