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Literature summary extracted from

  • Hilpert, K.; Wessner, H.; Schneider-Mergener, J.; Welfle, K.; Misselwitz, R.; Welfle, H.; Hocke, A.C.; Hippenstiel, S.; Hohne, W.
    Design and characterization of a hybrid miniprotein that specifically inhibits porcine pancreatic elastase (2003), J. Biol. Chem., 278, 24986-24993.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.21.36 EETI II trypsin-specific squash inhibitor from Ecballium elaterium Sus scrofa
3.4.21.36 HEI-TOE I hybrid inhibitor from Ecballium elaterium and the optimized binding loop of the third domain of turkey ovomucoid inhibitor Sus scrofa
3.4.21.36 HEI-TOE II
-
Sus scrofa
3.4.21.36 HEI-TOE III
-
Sus scrofa
3.4.21.36 MCEI III
-
Sus scrofa
3.4.21.36 OMTKY3 third Kazal-type domain of ovomucoid inhibitor from turkey egg white Sus scrofa
3.4.21.36 PACTLEYRC
-
Sus scrofa
3.4.21.36 PMTLEYR
-
Sus scrofa

Organism

EC Number Organism UniProt Comment Textmining
3.4.21.36 Sus scrofa P00772
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.21.36 succinyl-Ala-Ala-Phe-4-nitroanilide + H2O
-
Sus scrofa succinyl-Ala-Ala-Phe + 4-nitroaniline
-
?

Synonyms

EC Number Synonyms Comment Organism
3.4.21.36 PPE
-
Sus scrofa

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.4.21.36 0.000000024
-
OMTKY3 pH 8.5, 25°C Sus scrofa
3.4.21.36 0.000013
-
MCEI III pH 8.5, 25°C Sus scrofa
3.4.21.36 0.000049
-
PMTLEYR pH 5.5, 25°C Sus scrofa
3.4.21.36 0.000056
-
HEI-TOE III pH 8.5, 25°C Sus scrofa
3.4.21.36 0.00007
-
HEI-TOE II pH 8.5, 25°C Sus scrofa
3.4.21.36 0.000098
-
HEI-TOE I pH 8.5, 25°C Sus scrofa
3.4.21.36 0.00013
-
HEI-TOE I pH 6.5, 25°C Sus scrofa
3.4.21.36 0.00024
-
HEI-TOE III pH 5.0, 25°C Sus scrofa
3.4.21.36 0.00029
-
HEI-TOE III pH 7.5, 25°C Sus scrofa
3.4.21.36 0.00031
-
HEI-TOE III pH 6.5, 25°C Sus scrofa
3.4.21.36 0.00033
-
HEI-TOE I pH 5.5, 25°C Sus scrofa
3.4.21.36 0.00038
-
HEI-TOE I pH 7.5, 25°C Sus scrofa
3.4.21.36 0.00063
-
PMTLEYR pH 7.5, 25°C Sus scrofa
3.4.21.36 0.00067
-
PMTLEYR pH 8.5, 25°C Sus scrofa
3.4.21.36 0.0013
-
PMTLEYR pH 6.5, 25°C Sus scrofa
3.4.21.36 0.17
-
PACTLEYRC pH 8.5, 25°C Sus scrofa
3.4.21.36 0.82
-
EETI II pH 8.5, 25°C Sus scrofa