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Literature summary extracted from
- A new inhibitor design strategy for carboxypeptidase A as exemplified by N-(2-chloroethyl)-N-methylphenylalanine (2001), Bioorg. Med. Chem., 9, 237-243.
Inhibitors
| EC Number | Inhibitors | Comment | Organism | Structure |
|---|---|---|---|---|
| 3.4.17.1 | (R)-N-(2-chloroethyl)-N-methylphenylalanine | - |
Bos taurus |  |
| 3.4.17.1 | (S)-N-(2-chloroethyl)-N-methylphenylalanine | - |
Bos taurus | |
| 3.4.17.1 | rac-2-benzyl-5-chloropentanoic acid | - |
Bos taurus | |
Organism
| EC Number | Organism | UniProt | Comment | Textmining |
|---|---|---|---|---|
| 3.4.17.1 | Bos taurus | - |
- |
- |
Substrates and Products (Substrate)
| EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
|---|---|---|---|---|---|---|---|
| 3.4.17.1 | hippuryl-Phe + H2O | - |
Bos taurus | hippuric acid + Phe | - |
? | |
Ki Value [mM]
| EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
|---|---|---|---|---|---|---|
| 3.4.17.1 | 0.00036 | - |
(R)-N-(2-chloroethyl)-N-methylphenylalanine | pH 7.5 | Bos taurus | |
| 3.4.17.1 | 0.0016 | - |
rac-2-benzyl-5-chloropentanoic acid | pH 7.5 | Bos taurus | |
| 3.4.17.1 | 0.0025 | - |
(S)-N-(2-chloroethyl)-N-methylphenylalanine | pH 7.5 | Bos taurus | |
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Release 2023.1 (January 2023)
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