EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.B4 | alendronate | inhibits the in vitro invasion and random cell migration, 99% inhibition at 0.4 mM and physiological Ca2+-concentration, 67% inhibition at 0.4 mM and high Ca2+-concentration | Homo sapiens | |
3.4.24.B4 | clodronate | 77% inhibition at 0.4 mM and physiological Ca2+-concentration, 35.7% inhibition at 0.4 mM and high Ca2+-concentration | Homo sapiens | |
3.4.24.17 | alendronate | - |
Homo sapiens | |
3.4.24.17 | bisphosphonate | - |
Homo sapiens | |
3.4.24.17 | clodronate | - |
Homo sapiens | |
3.4.24.17 | pamidronate | - |
Homo sapiens | |
3.4.24.17 | zoledronate | - |
Homo sapiens |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.24.B4 | protein + H2O | Homo sapiens | - |
peptides | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.24.B4 | Homo sapiens | - |
- |
- |
3.4.24.17 | Homo sapiens | - |
human | - |
EC Number | Posttranslational Modification | Comment | Organism |
---|---|---|---|
3.4.24.B4 | proteolytic modification | autoactivation | Homo sapiens |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.24.B4 | C81-61 cell | melanoma cell line | Homo sapiens | - |
3.4.24.B4 | HT-1080 cell | fibrosaocoma cell line | Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.24.B4 | beta-casein + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.24.B4 | protein + H2O | - |
Homo sapiens | peptides | - |
? | |
3.4.24.17 | beta-casein + H2O | - |
Homo sapiens | ? | - |
? | |
3.4.24.17 | Fibronectin + H2O | - |
Homo sapiens | ? | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.24.B4 | M10.013 | Merops-ID | Homo sapiens |
3.4.24.B4 | matrix metalloproteinase-13 | - |
Homo sapiens |
3.4.24.B4 | MMP-13 | - |
Homo sapiens |
3.4.24.17 | MMP-3 | - |
Homo sapiens |
3.4.24.17 | stromelysin-1 | - |
Homo sapiens |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.24.B4 | 37 | - |
assay at | Homo sapiens |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.24.B4 | 7.8 | - |
assay at | Homo sapiens |