EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.22.51 | azocasein | substrate inhibition | Trypanosoma cruzi | |
3.4.22.51 | benzyloxycarbonyl-Phe-Arg-aminomethyl coumarin | substrate inhibition | Trypanosoma cruzi |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.22.51 | 0.003 | - |
benzyloxycarbonyl-Phe-Arg-aminomethyl coumarin | pH 4.5, 25°C | Trypanosoma cruzi | |
3.4.22.51 | 0.0032 | - |
benzyloxycarbonyl-Phe-Arg-aminomethyl coumarin | pH 8.5, 40°C | Trypanosoma cruzi | |
3.4.22.51 | 0.028 | - |
azocasein | pH 4.5, 25°C | Trypanosoma cruzi | |
3.4.22.51 | 0.029 | - |
azocasein | pH 8.5, 40°C | Trypanosoma cruzi |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.22.51 | Trypanosoma cruzi | Q598P5 | - |
- |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.22.51 | azocasein + H2O | - |
Trypanosoma cruzi | ? | - |
? | |
3.4.22.51 | benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Trypanosoma cruzi | ? | - |
? |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.22.51 | 0.023 | - |
benzyloxycarbonyl-Phe-Arg-aminomethyl coumarin | pH 4.5, 25°C | Trypanosoma cruzi | |
3.4.22.51 | 0.1 | - |
benzyloxycarbonyl-Phe-Arg-aminomethyl coumarin | pH 8.5, 40°C | Trypanosoma cruzi | |
3.4.22.51 | 0.48 | - |
azocasein | pH 8.5, 40°C | Trypanosoma cruzi | |
3.4.22.51 | 0.79 | - |
azocasein | pH 4.5, 25°C | Trypanosoma cruzi |