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Literature summary extracted from

  • Prade, L.; Engh, R.A.; Girod, A.; Kinzel, V.; Huber, R.; Bossemeyer, D.
    Staurosporine-induced conformational changes of cAMP-dependent protein kinase catalytic subunit explain inhibitory potential (1997), Structure, 5, 1627-1637.
    View publication on PubMed

Crystallization (Commentary)

EC Number Crystallization (Comment) Organism
2.7.11.11 crystal structure of the protein kinase catalytic subunit with staurosporine bound to the adenosine pocket Bos taurus

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.11.11 staurosporine
-
Bos taurus

Organism

EC Number Organism UniProt Comment Textmining
2.7.11.11 Bos taurus P00517
-
-

Synonyms

EC Number Synonyms Comment Organism
2.7.11.11 cAMP-dependent protein kinase, alpha-catalytic subunit
-
Bos taurus

Cofactor

EC Number Cofactor Comment Organism Structure
2.7.11.11 cAMP dependent on Bos taurus