EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
1.13.11.34 | adenosine | 58% of the activation with ATP | Homo sapiens | |
1.13.11.34 | ADP | 74% of the activation with ATP | Homo sapiens | |
1.13.11.34 | ADP-beta-S | 82% of the activation with ATP | Homo sapiens | |
1.13.11.34 | AMP | 68% of the activation with ATP | Homo sapiens | |
1.13.11.34 | AMP-4-nitrophenylphosphate | 77% of the activation with ATP | Homo sapiens | |
1.13.11.34 | ATP-alphaS | 118% of the activation with ATP | Homo sapiens | |
1.13.11.34 | ATP-gammaS | 80% of the activation with ATP | Homo sapiens |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
1.13.11.34 | L-670,630 | IC50: 0.0004 mM | Homo sapiens | |
1.13.11.34 | L-689,065 | IC50: 0.0003 mM | Homo sapiens | |
1.13.11.34 | L-697,198 | IC50: 0.00002 mM | Homo sapiens | |
1.13.11.34 | L-702,590 | - |
Homo sapiens | |
1.13.11.34 | L-702,701 | IC50: 0.0015 mM | Homo sapiens | |
1.13.11.34 | L705,302 | IC50: 0.00002 mM | Homo sapiens | |
1.13.11.34 | N-(4-chlorophenyl)-N-hydroxy-N'-(3-chlorophenyl)urea | IC50: 0.0001 mM | Homo sapiens | |
1.13.11.34 | ZD 2138 | i.e. CAS: 140841-32-3, IC50: 0.0003 mM | Homo sapiens | |
1.13.11.34 | zileuton | IC50: 0.01 | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
1.13.11.34 | Homo sapiens | - |
- |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
1.13.11.34 | recombinant enzyme | Homo sapiens |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
1.13.11.34 | arachidonate + O2 | i.e. 5,8,11,14-eicosatetraenoic acid | Homo sapiens | (6E,8Z,11Z,14Z)-(5S)-hydroperoxyicosa-6,8,11,14-tetraenoate | - |
? |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
1.13.11.34 | 0.00002 | - |
IC50: 0.00002 mM | Homo sapiens | L-697,198 | |
1.13.11.34 | 0.00002 | - |
IC50: 0.00002 mM | Homo sapiens | L705,302 | |
1.13.11.34 | 0.0001 | - |
IC50: 0.0001 mM | Homo sapiens | N-(4-chlorophenyl)-N-hydroxy-N'-(3-chlorophenyl)urea | |
1.13.11.34 | 0.0003 | - |
IC50: 0.0003 mM | Homo sapiens | L-689,065 | |
1.13.11.34 | 0.0003 | - |
i.e. CAS: 140841-32-3, IC50: 0.0003 mM | Homo sapiens | ZD 2138 | |
1.13.11.34 | 0.0004 | - |
IC50: 0.0004 mM | Homo sapiens | L-670,630 | |
1.13.11.34 | 0.0015 | - |
IC50: 0.0015 mM | Homo sapiens | L-702,701 | |
1.13.11.34 | 0.01 | - |
IC50: 0.01 mM | Homo sapiens | zileuton |