EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
1.14.99.1 | diclofenac | isozyme 1, 50% inhibition at 0.0003 mM, isozyme 2, 50% inhibition at 18 nM | Homo sapiens | |
1.14.99.1 | flurbiprofen | isozyme 1, 50% inhibition at 0.0009 mM, isozyme 2, 50% inhibition at 0.0009 mM | Homo sapiens | |
1.14.99.1 | Ibuprofen | isozyme 1, 50% inhibition at 0.009 mM, isozyme 2, 50% inhibition at 0.018 mM | Homo sapiens | |
1.14.99.1 | indomethacin | isozyme 1 50% inhibition at 0.0005 mM, isozyme 2, 50% inhibition at 0.0003 mM | Homo sapiens | |
1.14.99.1 | Ketoprofen | isozyme 1, 50% inhibition at 0.011 mM, isozyme 2, 50% inhibition at 0.018 mM | Homo sapiens | |
1.14.99.1 | L-745 | isozyme 1, 50% inhibition at 0.369 mM, isozyme 2, 50% inhibition at 0.002 mM | Homo sapiens | |
1.14.99.1 | meloxicam | isozyme 1, 50% inhibition at 0.005 mM, isozyme 2, 50% inhibition at 0.0004 mM | Homo sapiens | |
1.14.99.1 | N-[2-cyclohexyloxy-4-nitrophenyl]methanesulfonamide | isozyme 1, 50% inhibition at 0.017 mM, isozyme 2, 50% inhibition at 0.0001 mM | Homo sapiens | |
1.14.99.1 | nimesulide | isozyme 1, 50% inhibition at 0.009 mM, isozyme 2, 50% inhibition at 0.0005 mM | Homo sapiens | |
1.14.99.1 | piroxicam | isozyme 1, 50% inhibition at 0.009-0.024 mM, isozyme 2, 50% inhibition at 0.070-0.240 mM | Homo sapiens | |
1.14.99.1 | SC58125 | isozyme 1, 50% inhibition at 0.039 mM, isozyme 2, 50% inhibition at 0.0003 mM | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
1.14.99.1 | Homo sapiens | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
1.14.99.1 | monocyte | isozyme 2 | Homo sapiens | - |
1.14.99.1 | platelet | isozyme 1 | Homo sapiens | - |