EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.60 | 1,10-phenanthroline | metalloendopeptidase character | Homo sapiens | |
3.4.24.60 | benzamidine | weak | Homo sapiens | |
3.4.24.60 | EDTA | metalloendopeptidase character | Homo sapiens | |
3.4.24.60 | EGTA | metalloendopeptidase character | Homo sapiens | |
3.4.24.60 | additional information | no inhibition by N-tosyl-L-Phe chloromethyl ketone (i.e. TPCK); pepstatin, guanidylethylmercaptosuccinic acid (i.e. GEMSA), captopril, aprotinin, soybean trypsin inhibitor (i.e. STI), PMSF, IAA | Homo sapiens | |
3.4.24.60 | N-ethylmaleimide | - |
Homo sapiens | |
3.4.24.60 | p-chloromercuriphenylsulfonic acid | - |
Homo sapiens | |
3.4.24.60 | phosphoramidon | not | Homo sapiens | |
3.4.24.60 | thiorphan | not | Homo sapiens | |
3.4.24.60 | tosyl-Arg methyl ester | i.e. TAME, weak | Homo sapiens |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.60 | 0.019 | - |
atrial natriuretic peptide | - |
Homo sapiens |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
3.4.24.60 | extracellular | - |
Homo sapiens | - |
- |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.60 | additional information | metalloendopeptidase | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.24.60 | Homo sapiens | - |
- |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
3.4.24.60 | partial | Homo sapiens |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.24.60 | neuroblastoma cell line | NB-OK-1 | Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.24.60 | angiotensin II + H2O | i.e. Asp-Arg-Val-Tyr-Ile-His-Pro-Phe, cleavage site: Tyr4-Ile5 | Homo sapiens | ? | - |
? | |
3.4.24.60 | ANP-(103-126) + H2O | i.e. atrial natriuretic peptide, cleavage sites: Xaa-Phe, Xaa-Leu or Xaa-Ile bonds | Homo sapiens | ANP-(103-123) + Phe124-Arg125-Tyr126 | - |
? | |
3.4.24.60 | Asp-Ala-Asp-Thr-Cys-[D-Arg8]-kermit + H2O | model substrate, derivative of kermit, cleavage site: Ser12-Phe13 | Homo sapiens | ? | - |
? | |
3.4.24.60 | atrial natriuretic peptide + H2O | cleavage at Ser123-Phe124 | Homo sapiens | ? | - |
? | |
3.4.24.60 | bradykinin + H2O | i.e. Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg, major cleavage site: Gly4-Phe5, minor site: Pro7-Pro8 | Homo sapiens | ? | - |
? | |
3.4.24.60 | Litorin + H2O | minor sites: Gly6-His7 | Homo sapiens | ? | - |
? | |
3.4.24.60 | Litorin + H2O | major cleavage sites: His7-Phe8 | Homo sapiens | ? | - |
? | |
3.4.24.60 | additional information | no cleavage of analogous bonds in [Leu5]-enkephalin, oxytocin, vasopressin | Homo sapiens | ? | - |
? | |
3.4.24.60 | additional information | cleavage sites: Xaa-Phe, Xaa-Leu, Xaa-Ile | Homo sapiens | ? | - |
? | |
3.4.24.60 | Neuromedin C + H2O | Gly-Asn-His-Trp-Ala-Val-Gly-His-Leu-Met-NH2, major cleavage site: His8-Leu9, minor site: Gly7-His8 | Homo sapiens | ? | - |
? | |
3.4.24.60 | Somatostatin-14 + H2O | i.e. Ala-Gly-Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys, cleavage site: Phe6-Phe7 within disulfide bridged segment yielding one single product | Homo sapiens | ? | - |
? | |
3.4.24.60 | Substance P + H2O | major cleavage site: Gly9-Leu10, minor site: Phe7-Phe8 | Homo sapiens | ? | - |
? |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.24.60 | 7 | - |
- |
Homo sapiens |