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BRENDA support

Literature summary for 7.6.2.2 extracted from

  • Riccioni, R.; Dupuis, M.L.; Bernabei, M.; Petrucci, E.; Pasquini, L.; Mariani, G.; Cianfriglia, M.; Testa, U.
    The cancer stem cell selective inhibitor salinomycin is a p-glycoprotein inhibitor (2010), Blood Cells Mol. Dis., 45, 86-92.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
abamectin
-
Homo sapiens
nigericin
-
Homo sapiens
salinomycin treatment of the multidrug resistant cell lines with salinomycin restores a normal drug sensitivity of these cells Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
A-2780 cell multidrug resistant cancer cell line overexpressing P-gp Homo sapiens
-
CEM-VBL10 cell
-
Homo sapiens
-
CEM-VBL100 cell
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
multidrug resistance gp170
-
Homo sapiens