Inhibitors | Comment | Organism | Structure |
---|---|---|---|
orthovanadate | - |
Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Homo sapiens | 16020 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + asolectin/out | - |
Homo sapiens | ADP + phosphate + asolectin/in | - |
? | |
ATP + H2O + galactocerebroside/out | - |
Homo sapiens | ADP + phosphate + galactocerebroside/in | - |
? | |
ATP + H2O + lactocerebroside/out | - |
Homo sapiens | ADP + phosphate + lactocerebroside/in | - |
? | |
ATP + H2O + sphingomyelin/out | - |
Homo sapiens | ADP + phosphate + sphingomyelin/in | - |
? | |
ATP + H2O + verapamil/out | highest activity | Homo sapiens | ADP + phosphate + verapamil/in | - |
? | |
additional information | phosphatidylcholine, phosphatidylethanolamine, phophatidylserine, triglyceride, and cholesterol are no substrates of P-glycoprotein, ethyl acetate extracts from mouse brain homogenate exhibit weak substrate activity of P-glycoprotein | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ABCB1 | - |
Homo sapiens |
P-glycoprotein | - |
Homo sapiens |
P-gp | - |
Homo sapiens |