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Literature summary for 7.4.2.5 extracted from

  • Yang, B.; Hu, Y.; Smith, D.E.
    Impact of peptide transporter 1 on the intestinal absorption and pharmacokinetics of valacyclovir after oral dose escalation in wild-type and PepT1 knockout mice (2013), Drug Metab. Dispos., 41, 1867-1874.
    View publication on PubMedView publication on EuropePMC

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane
-
Mus musculus 16020
-

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
intestine
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + H2O + 5'-L-phenylalanyl-glycyl-floxuridine/in
-
Mus musculus ADP + phosphate + 5'-L-phenylalanyl-glycyl-floxuridine/out
-
?
ATP + H2O + midodrine/in
-
Mus musculus ADP + phosphate + midodrine/out
-
?
ATP + H2O + valacyclovir/in
-
Mus musculus ADP + phosphate + valacyclovir/out
-
?
ATP + H2O + valganciclovir/in
-
Mus musculus ADP + phosphate + valganciclovir /out
-
?

Synonyms

Synonyms Comment Organism
PepT1
-
Mus musculus
proton-coupled oligopeptide transporter 1
-
Mus musculus
solute carrier 15A1
-
Mus musculus