Activating Compound | Comment | Organism | Structure |
---|---|---|---|
8-pCPT-CGMP | induces a concentration-dependent increase in pump current, activator of PKG | Oryctolagus cuniculus | |
sodium nitroprusside | SNP, NO donor, not a simple concentration-dependent effect on pump current | Oryctolagus cuniculus | |
YC-1 | activator of soluble guanylyl cyclase, sGC | Oryctolagus cuniculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1H-[1,2,4]oxadiazole[4,3-a]quinoxalin-1-one | ODQ, inhibition of SNP-induced pump stimulation | Oryctolagus cuniculus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
sarcolemma | - |
Oryctolagus cuniculus | 42383 | - |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + phosphate + Na+/out | Oryctolagus cuniculus | - |
ATP + H2O + Na+/in | - |
? | |
ATP + H2O + K+/in | Oryctolagus cuniculus | - |
ADP + phosphate + K+/out | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
myocyte | ventricular myocyte | Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + phosphate + Na+/out | - |
Oryctolagus cuniculus | ATP + H2O + Na+/in | - |
? | |
ATP + H2O + K+/in | - |
Oryctolagus cuniculus | ADP + phosphate + K+/out | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Na+-K+ ATPase | - |
Oryctolagus cuniculus |
Na+-K+ pump | - |
Oryctolagus cuniculus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
2 | 8 | K+ | predicted, in the presence of 5.6 mM external K+ | Oryctolagus cuniculus | |
3 | 6 | K+ | predicted, in the presence of 15 mM external K+ | Oryctolagus cuniculus |