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Literature summary for 7.2.2.10 extracted from

  • Tatyanenko, L.V.; Khakina, E.A.; Zhilenkov, A.V.; Troshin, P.A.; Dobrokhotova, O.V.; Pikhteleva, I.Y.; Kotelnikov, A.I.
    Effects of fullerene derivatives on activity of Ca2+-ATPase of the sarcoplasmic reticulum and cGMP phosphodiesterase (2017), Bull. Exp. Biol. Med., 163, 321-325 .
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
polysubstituted fullerene C60-II noncompetitive and reversible inhibition, complete inhibition at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-III complete inhibition at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-IV 76% inhibition of Ca2+ transport and 91% inhibition of ATP hydrolysis at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-IX complete inhibition at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-V complete inhibition at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-VI 63% inhibition of Ca2+ transport and 38% inhibition of ATP hydrolysis at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-VII 60% inhibition of Ca2+ transport and 38% inhibition of ATP hydrolysis at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-VIII 82% inhibition of Ca2+ transport and 67% inhibition of ATP hydrolysis at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-X complete inhibition at 0.05 mM Oryctolagus cuniculus
polysubstituted fullerene C60-XI complete inhibition at 0.05 mM Oryctolagus cuniculus

Localization

Localization Comment Organism GeneOntology No. Textmining
sarcoplasmic reticulum
-
Oryctolagus cuniculus 16529
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + H2O + Ca2+[side 1] Oryctolagus cuniculus
-
ADP + phosphate + Ca2+[side 2]
-
?

Organism

Organism UniProt Comment Textmining
Oryctolagus cuniculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
muscle
-
Oryctolagus cuniculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + H2O + Ca2+[side 1]
-
Oryctolagus cuniculus ADP + phosphate + Ca2+[side 2]
-
?

Synonyms

Synonyms Comment Organism
Ca2+-ATPase
-
Oryctolagus cuniculus
sarcoplasmic reticulum Ca2+-ATPase
-
Oryctolagus cuniculus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0023
-
polysubstituted fullerene C60-II pH and temperature not specified in the publication Oryctolagus cuniculus