Inhibitors | Comment | Organism | Structure |
---|---|---|---|
rutin | - |
Oryctolagus cuniculus | |
rutin 4'''-O-arachidonate | - |
Oryctolagus cuniculus | |
rutin 4'''-O-erucate | - |
Oryctolagus cuniculus | |
rutin 4'''-O-linoleate | - |
Oryctolagus cuniculus | |
rutin 4'''-O-linolenate | - |
Oryctolagus cuniculus | |
rutin 4'''-O-oleate | - |
Oryctolagus cuniculus | |
rutin 4'''-O-stearate | - |
Oryctolagus cuniculus | |
rutin palmitate | - |
Oryctolagus cuniculus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
endoplasmic reticulum | - |
Oryctolagus cuniculus | 5783 | - |
sarcoplasmic reticulum | - |
Oryctolagus cuniculus | 16529 | - |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + Ca2+[side 1] | Oryctolagus cuniculus | - |
ADP + phosphate + Ca2+[side 2] | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | P04191 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
skeletal muscle | - |
Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + Ca2+[side 1] | - |
Oryctolagus cuniculus | ADP + phosphate + Ca2+[side 2] | - |
? |
Synonyms | Comment | Organism |
---|---|---|
sarcoplasmic reticulum calcium-dependent adenosine triphosphatase | - |
Oryctolagus cuniculus |
sarcoplasmic/endoplasmic reticulum Ca2+-ATPase | - |
Oryctolagus cuniculus |
SERCA1 | - |
Oryctolagus cuniculus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.023 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-arachidonate | |
0.025 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-linoleate | |
0.035 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-stearate | |
0.05 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-oleate | |
0.05 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-erucate | |
0.062 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin 4'''-O-linolenate | |
0.064 | - |
at 37°C and pH 7.4 | Oryctolagus cuniculus | rutin palmitate |